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On-target, dual aminopeptidase inhibition provides cross-species antimalarial activity by Edgar, RCS, Malcolm, TR, Siddiqui, G, Giannangelo, C, Counihan, NA, Challis, M, Duffy, S, Chowdhury, M, Marfurt, J, Dans, M, Wirjanata, G, Noviyanti, R, Daware, K, Suraweera, CD, Price, RN, Wittlin, S, Avery, VM, Drinkwater, N, Charman, SA, Creek, DJ, de Koning-Ward, TF, Scammells, PJ, McGowan, S
Published 2024Journal article -
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Hexahydroquinolines are antimalarial candidates with potent blood-stage and transmission-blocking activity by Vanaerschot, M, Lucantoni, L, Li, T, Combrinck, JM, Ruecker, A, Kumar, TRS, Rubiano, K, Ferreira, PE, Siciliano, G, Gulati, S, Henrich, PP, Ng, CL, Murithi, JM, Corey, VC, Duffy, S, Lieberman, OJ, Veiga, MI, Sinden, RE, Alano, P, Delves, MJ, Sim, K, Winzeler, EA, Egan, TJ, Hoffman, SL, Avery, VM, Fidock, DA
Published 2017Journal article -
3
3,3′-Disubstituted 5,5′-Bi(1,2,4-triazine) derivatives with potent in vitro and in vivo antimalarial activity by Xue, L, Shi, D-H, Harjani, JR, Huang, F, Beveridge, J, Dingjan, T, Ban, K, Diab, S, Duffy, S, Lucantoni, L, Fletcher, S, Chiu, FCK, Blundell, SA, Ellis, K, Ralph, SA, Wirjanata, G, Teguh, S, Noviyanti, R, Chavchich, M, Creek, DJ, Price, R, Marfurt, J, Charman, SA, Cuellar, M, Strasser, J, Dahlin, J, Walters, MA, Edstein, M, Avery, VM, Baell, JB
Published 2019Journal article