In silico tools to aid medicinal chemistry: optimising bromodomain inhibitors by Bluck, J

BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability by Jennings, L, Schiedel, M, Hewings, D, Picaud, S, Laurin, C, Bruno, P, Bluck, J, Scorah, A, See, L, Reynolds, J, Moroglu, M, Mistry, I, Hicks, A, Guzanov, P, Clayton, J, Evans, C, Stazi, G, Biggin, P, Mapp, A, Hammond, E, Humphreys, P, Filippakopoulos, P, Conway, S