Small-molecule inhibition of BRDT for male contraception. by Matzuk, M, McKeown, MR, Filippakopoulos, P, Li, Q, Ma, L, Agno, J, Lemieux, M, Picaud, S, Yu, R, Qi, J, Knapp, S, Bradner, J

Small-molecule bromodomain inhibitors for cancer therapy by Qi, J, Filippakopoulos, P, Picaud, S, Smith, W, Keates, T, Morse, E, Philpott, M, Shaw, K, Fedorov, O, West, N, Heightman, T, French, C, Knapp, S, Bradner, J

Click JAHAs: conformationally restricted ferrocene-based histone deacetylase inhibitors by Spencer, J, Amin, J, Boddiboyena, R, Packham, G, Cavell, B, Alwi, S, Paranal, R, Heightman, T, Wang, M, Marsden, B, Coxhead, P, Guille, M, Tizzard, G, Coles, S, Bradner, J

Click JAHAs: Conformationally restricted ferrocene-based histone deacetylase inhibitors by Spencer, J, Amin, J, Boddiboyena, R, Packham, G, Cavell, B, Syed Alwi, S, Paranal, R, Heightman, T, Wang, M, Marsden, B, Coxhead, P, Guille, M, Tizzard, G, Coles, S, Bradner, J

PFI-1, a highly selective protein interaction inhibitor, targeting BET Bromodomains. by Picaud, S, Da Costa, D, Thanasopoulou, A, Filippakopoulos, P, Fish, P, Philpott, M, Fedorov, O, Brennan, P, Bunnage, M, Owen, DR, Bradner, J, Taniere, P, O'Sullivan, B, Müller, S, Schwaller, J, Stankovic, T, Knapp, S

Selective inhibition of BET bromodomains. by Filippakopoulos, P, Qi, J, Picaud, S, Shen, Y, Smith, W, Fedorov, O, Morse, E, Keates, T, Hickman, T, Felletar, I, Philpott, M, Munro, S, McKeown, M, Wang, Y, Christie, A, West, N, Cameron, M, Schwartz, B, Heightman, T, La Thangue, N, French, C, Wiest, O, Kung, A, Knapp, S, Bradner, J

Selective inhibition of BET bromodomains. by Filippakopoulos, P, Qi, J, Picaud, S, Shen, Y, Smith, W, Fedorov, O, Morse, E, Keates, T, Hickman, T, Felletar, I, Philpott, M, Munro, S, McKeown, MR, Wang, Y, Christie, A, West, N, Cameron, M, Schwartz, B, Heightman, T, La Thangue, N, French, C, Wiest, O, Kung, A, Knapp, S, Bradner, J