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Kinetic and inhibition studies on human Jumonji-C (JmjC) domain-containing protein 5 by Tumber, A, Saleh, E, Brewitz, L, Corner, TP, Schofield, CJ
Published 2023Journal article -
2
5-substituted pyridine-2,4-dicarboxylate derivatives have potential for selective inhibition of human Jumonji-C domain-containing protein 5 by Brewitz, L, Nakashima, Y, Piasecka, SK, Salah, E, Fletcher, SC, Tumber, A, Corner, TP, Kennedy, TJ, Fiorini, G, Thalhammer, A, Christensen, KE, Coleman, ML, Schofield, CJ
Published 2023Journal article -
3
Structure-guided optimisation of N-hydroxythiazole-derived inhibitors of factor inhibiting hypoxia-inducible factor-α by Corner, TP, Teo, RZR, Wu, Y, Salah, E, Nakashima, Y, Fiorini, G, Tumber, A, Brasnett, A, Holt-Martyn, JP, Figg, WD, Zhang, X, Brewitz, L, Schofield, CJ
Published 2023Journal article