The first Pd-catalyzed Buchwald–Hartwig aminations at C-2 or C-4 in the estrone series by Ildikó Bacsa, Dávid Szemerédi, János Wölfling, Gyula Schneider, Lilla Fekete, Erzsébet Mernyák

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Synthesis of substituted 15β-alkoxy estrone derivatives and their cofactor-dependent inhibitory effect on 17β-HSD1 by Bianka Edina Herman, Anita Kiss, János Wölfling, Erzsébet Mernyák, Mihály Szécsi, Gyula Schneider

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Electrophile- and Lewis acid-induced nitrone formation and 1,3-dpolar cycloaddition reactions in the 13α- and 13β-estrone series by Erzsebet Mernyak, Judit Huber, Gabriella Benedek, Roland Pfoh, Stephan Rühl, Gyula Schneider, János Wölfling

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Synthesis of novel 13α-estrone derivatives by Sonogashira coupling as potential 17β-HSD1 inhibitors by Ildikó Bacsa, Rebeka Jójárt, János Wölfling, Gyula Schneider, Bianka Edina Herman, Mihály Szécsi, Erzsébet Mernyák

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Synthesis of Novel C-2- or C-15-Labeled BODIPY—Estrone Conjugates by Ildikó Bacsa, Csilla Konc, Anna Boglárka Orosz, Gábor Kecskeméti, Réka Rigó, Csilla Özvegy-Laczka, Erzsébet Mernyák

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Synthesis and in Vitro Antiproliferative Evaluation of C-13 Epimers of Triazolyl-d-Secoestrone Alcohols: The First Potent 13α-d-Secoestrone Derivative by Johanna Szabó, Nóra Jerkovics, Gyula Schneider, János Wölfling, Noémi Bózsity, Renáta Minorics, István Zupkó, Erzsébet Mernyák

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Pd-Catalyzed microwave-assisted synthesis of phosphonated 13α-estrones as potential OATP2B1, 17β-HSD1 and/or STS inhibitors by Rebeka Jójárt, Szabolcs Pécsy, György Keglevich, Mihály Szécsi, Réka Rigó, Csilla Özvegy-Laczka, Gábor Kecskeméti, Erzsébet Mernyák

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Synthesis, Biological Evaluation and Docking Studies of 13-Epimeric 10-fluoro- and 10-Chloroestra-1,4-dien-3-ones as Potential Aromatase Inhibitors by Rebeka Jójárt, Péter Traj, Édua Kovács, Ágnes Horváth, Gyula Schneider, Mihály Szécsi, Attila Pál, Gábor Paragi, Erzsébet Mernyák

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Synthesis and Antiproliferative Activity of Steroidal Diaryl Ethers by Édua Kovács, Hazhmat Ali, Renáta Minorics, Péter Traj, Vivien Resch, Gábor Paragi, Bella Bruszel, István Zupkó, Erzsébet Mernyák

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Transition metal-catalysed A-ring C–H activations and C(sp2)–C(sp2) couplings in the 13α-oestrone series and in vitro evaluation of antiproliferative properties by Péter Traj, Ali Hazhmat Abdolkhaliq, Anett Németh, Sámuel Trisztán Dajcs, Ferenc Tömösi, Tea Lanisnik-Rizner, István Zupkó, Erzsébet Mernyák

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Investigation of the Antineoplastic Effects of 2-(4-Chlorophenyl)-13α-Estrone Sulfamate against the HPV16-Positive Human Invasive Cervical Carcinoma Cell Line SiHa by Hazhmat Ali, Péter Traj, Gábor J. Szebeni, Nikolett Gémes, Vivien Resch, Gábor Paragi, Erzsébet Mernyák, Renáta Minorics, István Zupkó

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Synthesis and evaluation of anticancer activities of 2- or 4-substituted 3-(N-benzyltriazolylmethyl)-13α-oestrone derivatives by Rebeka Jójárt, Seyyed Ashkan Senobar Tahaei, Péter Trungel-Nagy, Zoltán Kele, Renáta Minorics, Gábor Paragi, István Zupkó, Erzsébet Mernyák

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Synthesis and Biological Evaluation of Triazolyl 13α-Estrone–Nucleoside Bioconjugates by Brigitta Bodnár, Erzsébet Mernyák, János Wölfling, Gyula Schneider, Bianka Edina Herman, Mihály Szécsi, Izabella Sinka, István Zupkó, Zoltán Kupihár, Lajos Kovács

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Microwave-assisted Phospha-Michael addition reactions in the 13α-oestrone series and in vitro antiproliferative properties by Erzsébet Mernyák, Sándor Bartha, Lili Kóczán, Rebeka Jójárt, Vivien Resch, Gábor Paragi, Máté Vágvölgyi, Attila Hunyadi, Bella Bruszel, István Zupkó, Renáta Minorics

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Antiproliferative and Antimetastatic Properties of 16-Azidomethyl Substituted 3-<i>O</i>-Benzyl Estrone Analogs by Seyyed Ashkan Senobar Tahaei, Ágnes Kulmány, Renáta Minorics, Anita Kiss, Zoltán Szabó, Péter Germán, Gábor J. Szebeni, Nikolett Gémes, Erzsébet Mernyák, István Zupkó

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Synthesis and structure–activity relationships of 2- and/or 4-halogenated 13β- and 13α-estrone derivatives as enzyme inhibitors of estrogen biosynthesis by Ildikó Bacsa, Bianka Edina Herman, Rebeka Jójárt, Kevin Stefán Herman, János Wölfling, Gyula Schneider, Mónika Varga, Csaba Tömböly, Tea Lanišnik Rižner, Mihály Szécsi, Erzsébet Mernyák

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