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Amino Acid Replacement at Position 228 Induces Fluctuation in the Ω-Loop of KPC-3 and Reduces the Affinity against Oxyimino Cephalosporins: Kinetic and Molecular Dynamics Studies by Alessandra Piccirilli, Fabrizia Brisdelli, Jean Denis Docquier, Massimiliano Aschi, Sabrina Cherubini, Filomena De Luca, André Matagne, Gianfranco Amicosante, Mariagrazia Perilli
Published 2020-12-01
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Optimization of Pyrazole Compounds as Antibiotic Adjuvants Active against Colistin- and Carbapenem-Resistant <i>Acinetobacter baumannii</i> by Filomena Sannio, Antonella Brizzi, Rosita Del Prete, Marialuce Avigliano, Tiziana Simone, Carlotta Pagli, Teresa Ferraro, Filomena De Luca, Marco Paolino, Federico Corelli, Claudia Mugnaini, Jean-Denis Docquier
Published 2022-12-01
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4-(<i>N</i>-Alkyl- and -Acyl-amino)-1,2,4-triazole-3-thione Analogs as Metallo-β-Lactamase Inhibitors: Impact of 4-Linker on Potency and Spectrum of Inhibition by Laurent Gavara, Federica Verdirosa, Alice Legru, Paola Sandra Mercuri, Lionel Nauton, Laurent Sevaille, Georges Feller, Dorothée Berthomieu, Filomena Sannio, Francesca Marcoccia, Silvia Tanfoni, Filomena De Luca, Nohad Gresh, Moreno Galleni, Jean-Denis Docquier, Jean-François Hernandez
Published 2020-07-01
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