The Zinc-Sensing Receptor GPR39 in Physiology and as a Pharmacological Target by Anna Laitakari, Lingzhi Liu, Thomas M. Frimurer, Birgitte Holst

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Assessment and challenges of ligand docking into comparative models of G-protein coupled receptors. by Elizabeth Dong Nguyen, Christoffer Norn, Thomas M Frimurer, Jens Meiler

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Receptor structure-based discovery of non-metabolite agonists for the succinate receptor GPR91 by Trauelsen, M, Ulven, E, Hjorth, SA, Brvar, M, Monaco, C, Frimurer, TM, Schwartz, TW

H4K20me0 recognition by BRCA1–BARD1 directs homologous recombination to sister chromatids by Nakamura, K, Saredi, G, Becker, J, Foster, B, Nguyen, N, Beyer, T, Cesa, L, Faull, P, Lukauskas, S, Frimurer, T, Chapman, J, Bartke, T, Groth, A

Extracellular succinate hyperpolarizes M2 macrophages through SUCNR1/GPR91-mediated Gq signaling by Mette Trauelsen, Thomas K. Hiron, Da Lin, Jacob E. Petersen, Billy Breton, Anna Sofie Husted, Siv A. Hjorth, Asuka Inoue, Thomas M. Frimurer, Michel Bouvier, Chris A. O’Callaghan, Thue W. Schwartz

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Human substance P receptor binding mode of the antagonist drug aprepitant by NMR and crystallography by Shuanghong Chen, Mengjie Lu, Dongsheng Liu, Lingyun Yang, Cuiying Yi, Limin Ma, Hui Zhang, Qing Liu, Thomas M. Frimurer, Ming-Wei Wang, Thue W. Schwartz, Raymond C. Stevens, Beili Wu, Kurt Wüthrich, Qiang Zhao

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Selective release of gastrointestinal hormones induced by an orally active GPR39 agonist by Kaare V. Grunddal, Thi A. Diep, Natalia Petersen, Iain R. Tough, Louise J. Skov, Lingzhi Liu, Jesse A. Buijink, Franziska Mende, Chunyu Jin, Sara L. Jepsen, Louis M.E. Sørensen, Michael P. Achiam, Rune B. Strandby, Anders Bach, Bolette Hartmann, Thomas M. Frimurer, Siv A. Hjorth, Michel Bouvier, Helen Cox, Birgitte Holst

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