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Identification of a chemical probe for family VIII bromodomains through optimization of a fragment hit by Gerstenberger, BS, Trzupek, JD, Tallant, C, Fedorov, O, Filippakopoulos, P, Brennan, PE, Fedele, V, Martin, S, Picaud, S, Rogers, C, Parikh, M, Taylor, A, Samas, B, O'Mahony, A, Berg, E, Pallares, G, Torrey, AD, Treiber, DK, Samardjiev, IJ, Nasipak, BT, Padilla-Benavides, T, Wu, Q, Imbalzano, AN, Nickerson, JA, Bunnage, ME, Müller, S, Knapp, S, Owen, DR
Published 2016Journal article -
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Selective targeting of bromodomains of the bromodomain-PHD fingers family impairs osteoclast differentiation by Meier, JC, Tallant, C, Fedorov, O, Witwicka, H, Hwang, SY, van Stiphout, RG, Lambert, JP, Rogers, C, Yapp, C, Gerstenberger, BS, Fedele, V, Savitsky, P, Heidenreich, D, Daniels, DL, Owen, DR, Fish, PV, Igoe, NM, Bayle, ED, Haendler, B, Oppermann, UCT, Buffa, F, Brennan, PE, Müller, S, Gingras, AC, Odgren, PR, Birnbaum, MJ, Knapp, S
Published 2017Journal article