ERAP1 inhibitor development by Guzanov, P

BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability by Jennings, L, Schiedel, M, Hewings, D, Picaud, S, Laurin, C, Bruno, P, Bluck, J, Scorah, A, See, L, Reynolds, J, Moroglu, M, Mistry, I, Hicks, A, Guzanov, P, Clayton, J, Evans, C, Stazi, G, Biggin, P, Mapp, A, Hammond, E, Humphreys, P, Filippakopoulos, P, Conway, S