Evaluation of Potency of Known Oximes (Pralidoxime, Trimedoxime, HI-6, Methoxime, Obidoxime) to in vitro Reactivate Acetylcholinesterase Inhibited by Pesticides (Chlorpyrifos and M... by Kamil Musílek, Kamil Kuča, Daniel Jun

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Novel Group of AChE Reactivators—Synthesis, In Vitro Reactivation and Molecular Docking Study by David Malinak, Eugenie Nepovimova, Daniel Jun, Kamil Musilek, Kamil Kuca

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C‑3 Steroidal Hemiesters as Inhibitors of 17β-Hydroxysteroid Dehydrogenase Type 10 by Michaela Hanzlova, Barbora Slavikova, Marina Morozovova, Kamil Musilek, Aneta Rotterova, Lucie Zemanová, Eva Kudova

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Correction to “C‑3 Steroidal Hemiesters as Inhibitors of 17β-Hydroxysteroid Dehydrogenase Type 10” by Michaela Hanzlova, Barbora Slavikova, Marina Morozovova, Kamil Musilek, Aneta Rotterova, Lucie Zemanová, Eva Kudova

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Targeted Synthesis of 1-(4-Hydroxyiminomethylpyridinium)-3-pyridiniumpropane Dibromide – A New Nerve Agent Reactivator by Jan Marek, Martina Hrabinova, Petr Stodulka, Daniel Jun, Martin Paar, Kamil Musilek, Kamil Kuca

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Preparation of Benzalkonium Salts Differing in the Length of a Side Alkyl Chain by Daniel Jun, Martina Hrabinova, Petra Hanusova, Kamil Musilek, Petr Stodulka, Jan Marek, Kamil Kuca

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Molecular Modeling Studies on the Multistep Reactivation Process of Organophosphate-Inhibited Acetylcholinesterase and Butyrylcholinesterase by Jakub Jończyk, Jędrzej Kukułowicz, Kamil Łątka, Barbara Malawska, Young-Sik Jung, Kamil Musilek, Marek Bajda

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1,2,4-Triazole-based anticonvulsant agents with additional ROS scavenging activity are effective in a model of pharmacoresistant epilepsy by Barbara Kaproń, Robert Czarnomysy, Mariusz Wysokiński, Rudolf Andrys, Kamil Musilek, Andrea Angeli, Claudiu T. Supuran, Tomasz Plech

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Preparation of the Pyridinium Salts Differing in the Length of the N-Alkyl Substituent by Kamil Musilek, Jan Korabecny, Miroslav Pohanka, Ondrej Soukup, Jiri Cabal, Petr Stodulka, Jan Marek, Kamil Kuca

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Charged pyridinium oximes with thiocarboxamide moiety are equally or less effective reactivators of organophosphate-inhibited cholinesterases compared to analogous carboxamides by Zuzana Kohoutova, David Malinak, Rudolf Andrys, Jana Svobodova, Miroslav Psotka, Monika Schmidt, Lukas Prchal, Kamil Musilek

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Preparation of Quinolinium Salts Differing in the Length of the Alkyl Side Chain by Kamil Kuca, Kallol K. Ghosh, Kamil Musilek, Jiri Cabal, Petr Stodulka, Ondrej Soukup, Vladimir Buchta, Jan Marek

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Molecular Modeling Studies on the Interactions of Aflatoxin B1 and Its Metabolites with Human Acetylcholinesterase. Part II: Interactions with the Catalytic Anionic Site (CAS) by Joyce S. F. D. de Almeida, Rafael Dolezal, Ondrej Krejcar, Kamil Kuca, Kamil Musilek, Daniel Jun, Tanos C. C. França

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Anticipated Social and Healthcare Economic Burden of People with Alzheimer’s Disease in Two Selected Regions of the Czech Republic by Petra Maresova, Lenka Komarkova, Jitka Kuhnova, Richard Cimler, Peter Pazitny, Daniela Kandilaki, Kamil Musilek, Zuzana Truhlarova, Filip Zemek, Kamil Kuca

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7-Methoxytacrine-Adamantylamine Heterodimers as Cholinesterase Inhibitors in Alzheimer’s Disease Treatment — Synthesis, Biological Evaluation and Molecular Modeling Studies by Kamil Kuca, Katarina Siposova, Lucie Drtinova, Zuzana Gazova, Ondrej Soukup, Kamil Musilek, Anna Horova, Katarina Spilovska, Jan Korabecny, Jan Kral

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Novel Bisquaternary Oximes—Reactivation of Acetylcholinesterase and Butyrylcholinesterase Inhibited by Paraoxon by Daniel Jun, Jana Zdarova Karasova, Miroslav Pohanka, Martina Hrabinova, Kamil Musilek, Martin Paar, Vladimir Cirkva, Jiri Palecek, Kamil Kuca, Lucie Musilova

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BODIPY-labelled acetylcholinesterase reactivators can be encapsulated into ferritin nanovehicles for enhanced bioavailability in the CNS by Eliska Prchalova, Martina Sukupova, David Malinak, Rudolf Andrys, Ladislav Sivak, Vladimir Pekarik, Adam Skarka, Jana Svobodova, Lukas Prchal, Lukas Fresser, Zbynek Heger, Kamil Musilek

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1-(Benzo[d]thiazol-2-yl)-3-phenylureas as dual inhibitors of casein kinase 1 and ABAD enzymes for treatment of neurodegenerative disorders by Ondrej Benek, Lukas Hroch, Laura Aitken, Frank Gunn-Moore, Lucie Vinklarova, Kamil Kuca, Daniel I. Perez, Concepcion Perez, Ana Martinez, Zdenek Fisar, Kamil Musilek

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Synthesis, Biological Evaluation, and Docking Studies of Novel Bisquaternary Aldoxime Reactivators on Acetylcholinesterase and Butyrylcholinesterase Inhibited by Paraoxon by Kamil Kuca, Daniel Jun, Lucie Junova, Kamil Musilek, Martina Hrabinova, Jorge Alberto Valle da Silva, Teodorico Castro Ramalho, Marian Valko, Qinghua Wu, Eugenie Nepovimova, Tanos Celmar Costa França

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Donepezil + chromone + melatonin hybrids as promising agents for Alzheimer’s disease therapy by Irene Pachón-Angona, Bernard Refouvelet, Rudolf Andrýs, Helène Martin, Vincent Luzet, Isabel Iriepa, Ignacio Moraleda, Daniel Diez-Iriepa, María-Jesús Oset-Gasque, José Marco-Contelles, Kamil Musilek, Lhassane Ismaili

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Synthesis and In Vitro Evaluation of Novel Dopamine Receptor D₂ 3,4-dihydroquinolin-2(1<i>H</i>)-one Derivatives Related to Aripiprazole by Radomir Juza, Kristyna Stefkova, Wim Dehaen, Alena Randakova, Tomas Petrasek, Iveta Vojtechova, Tereza Kobrlova, Lenka Pulkrabkova, Lubica Muckova, Marko Mecava, Lukas Prchal, Eva Mezeiova, Kamil Musilek, Ondrej Soukup, Jan Korabecny

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