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A triazolopyrimidine-based dihydroorotate dehydrogenase inhibitor (DSM421) with improved drug-like properties for treatment and prevention of malaria by Phillips, M, White, K, Kokkonda, S, Deng, X, White, J, El Mazouni, F, Marsh, K, Tomchick, D, Manjalanagara, K, Rudra, K, Wirjanata, G, Noviyanti, R, Price, R, Marfurt, J, Shackleford, D, Chiu, F, Campbell, M, Jimenez Diaz, M, Ferrer-Bazaga, S, Angulo-Barturen, I, Martínez-Martínez, M, Lafuente-Monasterio, M, Kaminsky, W, Silue, K, Zeeman, A, Kocken, C, Leroy, D, Blasco, B, Rossignol, E, Rueckle, T, Matthews, D, Burrows, J, Waterson, D, Palmer, M, Rathod, P, Charman, S
Published 2016Journal article -
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Open Source Drug Discovery: Highly Potent Antimalarial Compounds Derived from the Tres Cantos Arylpyrroles. by Williamson, A, Ylioja, P, Robertson, M, Antonova-Koch, Y, Avery, V, Baell, J, Batchu, H, Batra, S, Burrows, J, Bhattacharyya, S, Calderon, F, Charman, S, Clark, J, Crespo, B, Dean, M, Debbert, S, Delves, M, Dennis, A, Deroose, F, Duffy, S, Fletcher, S, Giaever, G, Hallyburton, I, Gamo, F, Gebbia, M, Guy, R, Hungerford, Z, Kirk, K, Lafuente-Monasterio, M, Lee, A, Meister, S, Nislow, C, Overington, J, Papadatos, G, Patiny, L, Pham, J, Ralph, S, Ruecker, A, Ryan, E, Southan, C, Srivastava, K, Swain, C, Tarnowski, M, Thomson, P, Turner, P, Wallace, I, Wells, T, White, K, White, L, Willis, P, Winzeler, E, Wittlin, S, Todd, M
Published 2016Journal article