Structural characterization of human Vaccinia-Related Kinases (VRK) bound to small-molecule inhibitors identifies different P-loop conformations by Couñago, R, Allerston, C, Savitsky, P, Azevedo, H, Godoi, P, Wells, C, Mascarello, A, de Souza Gama, F, Massirer, K, Zuercher, W, Guimarães, C, Gileadi, O

Quinoxaline-substituted chalcones as new inhibitors of breast cancer resistance protein ABCG2: polyspecificity at B-ring position by Winter E, Gozzi GJ, Chiaradia-Delatorre LD, Daflon-Yunes N, Terreux R, Gauthier C, Mascarello A, Leal PC, Cadena SM, Yunes RA, Nunes RJ, Creczynski-Pasa TB, Di Pietro A

Get full text

Development of pyridine-based inhibitors for the human vaccinia-related kinases 1 and 2 by Serafim, R, De Souza Gama, F, Dutra, L, Dos Reis, C, Vasconcelos, S, Da Silva Santiago, A, Takarada, J, Di Pillo, F, Azevedo, H, Mascarello, A, Elkins, J, Massirer, K, Gileadi, O, Guimarães, C, Couñago, R