Structure-based bioisosteric design, synthesis and biological evaluation of novel pyrimidines as antiplasmodial antifolate agents by Moaz M. Abdou, Paul M. O'Neill, Eric Amigues, Magdalini Matziari

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Unprecedented Convergent Synthesis of Sugar-Functionalization of Phosphinic Acids under Metal-Free Conditions by Moaz M. Abdou, Paul M. O’Neill, Eric Amigues, Magdalini Matziari

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Antimalarial Agents as Therapeutic Tools Against Toxoplasmosis—A Short Bridge between Two Distant Illnesses by Alina Secrieru, Inês C. C. Costa, Paul M. O'Neill, Maria L. S. Cristiano

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Diastereoselective synthesis of a novel phosphinic peptide as ACE inhibitor: Fragment-based design approach by Moaz M. Abdou, Dewen Dong, Paul M. O'Neill, Eric Amigues, Magdalini Matziari

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Ebselen analogues delay disease onset and its course in fALS by on-target SOD-1 engagement by Seiji Watanabe, Kangsa Amporndanai, Raheela Awais, Caroline Latham, Muhammad Awais, Paul M. O’Neill, Koji Yamanaka, S. Samar Hasnain

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X-ray and cryo-EM structures of inhibitor-bound cytochrome bc1 complexes for structure-based drug discovery by Kangsa Amporndanai, Rachel M. Johnson, Paul M. O'Neill, Colin W. G. Fishwick, Alexander H. Jamson, Shaun Rawson, Stephen P. Muench, S. Samar Hasnain, Svetlana V. Antonyuk

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Targeting the Ubiquinol-Reduction (Q_i) Site of the Mitochondrial Cytochrome <i>bc₁</i> Complex for the Development of Next Generation Quinolone Antimalarials by Kangsa Amporndanai, Nattapon Pinthong, Paul M. O’Neill, W. David Hong, Richard K. Amewu, Chandrakala Pidathala, Neil G. Berry, Suet C. Leung, Stephen A. Ward, Giancarlo A. Biagini, S. Samar Hasnain, Svetlana V. Antonyuk

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Optimizing drug discovery for snakebite envenoming via a high-throughput phospholipase A2 screening platform by Laura-Oana Albulescu, Laura-Oana Albulescu, Adam Westhorpe, Adam Westhorpe, Rachel H. Clare, Rachel H. Clare, Christopher M. Woodley, Nivya James, Jeroen Kool, Neil G. Berry, Paul M. O’Neill, Nicholas R. Casewell, Nicholas R. Casewell

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Snakebite drug discovery: high-throughput screening to identify novel snake venom metalloproteinase toxin inhibitors by Rachel H. Clare, Rachel H. Clare, Charlotte A. Dawson, Charlotte A. Dawson, Adam Westhorpe, Adam Westhorpe, Laura-Oana Albulescu, Laura-Oana Albulescu, Christopher M. Woodley, Nada Mosallam, Daniel J. W. Chong, Jeroen Kool, Neil G. Berry, Paul M. O’Neill, Nicholas R. Casewell, Nicholas R. Casewell

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