Linkers as Game-changers in PROTAC Technology: Emphasizing General Trends in PROTAC Pharmacokinetics for their Rational Design by Carlotta Cecchini, Sébastien Tardy, Leonardo Scapozza

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From Conception to Development: Investigating PROTACs Features for Improved Cell Permeability and Successful Protein Degradation by Carlotta Cecchini, Carlotta Cecchini, Sara Pannilunghi, Sara Pannilunghi, Sébastien Tardy, Sébastien Tardy, Leonardo Scapozza, Leonardo Scapozza

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Exploring the Ubiquitin-Proteasome System (UPS) through PROTAC Technology by Carlotta Cecchini, Sébastien Tardy, Valentina Ceserani, Jean-Philippe Theurillat, Leonardo Scapozza

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Novel Mechanism for an Old Drug: Phenazopyridine is a Kinase Inhibitor Affecting Autophagy and Cellular Differentiation by Olivier Preynat-Seauve, Olivier Preynat-Seauve, Evelyne Bao-Vi Nguyen, Yvonne Westermaier, Margaux Héritier, Sébastien Tardy, Yves Cambet, Maxime Feyeux, Aurélie Caillon, Leonardo Scapozza, Karl-Heinz Krause, Karl-Heinz Krause

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Isolation and Identification of Isocoumarin Derivatives With Specific Inhibitory Activity Against Wnt Pathway and Metabolome Characterization of Lasiodiplodia venezuelensis by Léonie Pellissier, Léonie Pellissier, Alexey Koval, Laurence Marcourt, Laurence Marcourt, Emerson Ferreira Queiroz, Emerson Ferreira Queiroz, Nicole Lecoultre, Sara Leoni, Luis-Manuel Quiros-Guerrero, Luis-Manuel Quiros-Guerrero, Morgane Barthélémy, Bastiaan L. Duivelshof, Bastiaan L. Duivelshof, Davy Guillarme, Davy Guillarme, Sébastien Tardy, Sébastien Tardy, Véronique Eparvier, Karl Perron, Karl Perron, Jérôme Chave, Didier Stien, Katia Gindro, Vladimir Katanaev, Vladimir Katanaev, Jean-Luc Wolfender, Jean-Luc Wolfender

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Correction to “Discovery of Novel α‑Carboline Inhibitors of the Anaplastic Lymphoma Kinase” by Luca Mologni, Sébastien Tardy, Alfonso Zambon, Alexandre Orsato, Cédric Schneider, William H. Bisson, Monica Ceccon, Michela Viltadi, David Goyard, Pierre Garcia, Joseph D’Attoma, Sara Pannilunghi, Vito Vece, Jerome Bertho, David Gueyrard, Peter Goekjian, Leonardo Scapozza, Carlo Gambacorti-Passerini

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