A high-throughput small molecule screen identifies synergism between DNA methylation and Aurora kinase pathways for X reactivation by Lessing, Derek, Dial, Thomas O., Wei, Chunyao, Payer, Bernhard, Carrette, Lieselot L. G., Kesner, Barry, Szanto, Attila, Jadhav, Ajit, Maloney, David J., Simeonov, Anton, Theriault, Jimmy, Hasaka, Thomas, Bedalov, Antonio, Bartolomei, Marisa S., Lee, Jeannie T.

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Discovery and optimization of piperazine-1-thiourea-based human phosphoglycerate dehydrogenase inhibitors by Rohde, Jason M., Brimacombe, Kyle R., Liu, Li, Pacold, Michael Edward, Yasgar, Adam, Cheff, Dorian M., Lee, Tobie D., Rai, Ganesha, Baljinnyam, Bolormaa, Li, Zhuyin, Simeonov, Anton, Hall, Matthew D., Shen, Min, Sabatini, David, Boxer, Matthew B.

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