Showing 1 - 6 results of 6 for search 'Szommer, T', query time: 0.03s
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Novel Starting Points for Human Glycolate Oxidase Inhibitors, Revealed by Crystallography-Based Fragment Screening by Sabrina R. Mackinnon, Gustavo A. Bezerra, Tobias Krojer, Tamas Szommer, Tamas Szommer, Frank von Delft, Frank von Delft, Paul E. Brennan, Paul E. Brennan, Wyatt W. Yue
Published 2022-05-01
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Inhibition of histone H3K27 demethylases inactivates brachyury (TBXT) and promotes chordoma cell death by Cottone, L, Cribbs, AP, Khandelwal, G, Wells, G, Ligammari, L, Philpott, M, Tumber, A, Lombard, P, Hookway, ES, Szommer, T, Johansson, C, Brennan, PE, Pillay, N, Jenner, RG, Oppermann, U, Flanagan, AM
Published 2020Journal article -
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Discovery of a highly selective cell‐active inhibitor of the histone lysine demethylases KDM2/7 by Gerken, P, Wolstenhume, J, Tumbler, A, Hatch, S, Zhang, Y, Muller, S, Chandler, S, Mair, B, Li, F, Nijman, S, Konietzny, R, Szommer, T, Yapp, C, Fedorov, O, Benesch, J, Vedadi, M, Kessler, B, Kawamura, A, Brennan, P, Smith, M
Published 2017Journal article -
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Discovery of a highly selective cell-active inhibitor of the histone lysine demethylases KDM2/7 by Gerken, PA, Wolstenhulme, JR, Tumber, AM, Hatch, SB, Zhang, Y, Müller, S, Chandler, SA, Mair, B, Li, F, Nijman, SMB, Konietzny, R, Szommer, T, Yapp, C, Fedorov, O, Benesch, JLP, Vedadi, M, Kessler, BM, Kawamura, A, Brennan, PE, Smith, MD
Published 2017Journal article -
5
Unexpected Noncovalent Off-Target Activity of Clinical BTK Inhibitors Leads to Discovery of a Dual NUDT5/14 Antagonist by Balıkçı, E, Marques, AMC, Bauer, LG, Seupel, R, Bennett, J, Raux, B, Buchan, K, Simelis, K, Singh, U, Rogers, C, Ward, J, Cheng, C, Szommer, T, Schützenhofer, K, Elkins, JM, Sloman, DL, Ahel, I, Fedorov, O, Brennan, PE, Huber, KVM
Published 2024Journal article -
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Rapid covalent-probe discovery by electrophile-fragment screening by Resnick, E, Bradley, A, Gan, J, Douangamath, A, Krojer, T, Sethi, R, Geurink, PP, Aimon, A, Amitai, G, Bellini, D, Bennett, J, Fairhead, M, Fedorov, O, Gabizon, R, Gan, J, Guo, J, Plotnikov, A, Reznik, N, Ruda, GF, Díaz-Sáez, L, Straub, VM, Szommer, T, Velupillai, S, Zaidman, D, Zhang, Y, Coker, AR, Dowson, CG, Barr, HM, Wang, C, Huber, KVM, Brennan, PE, Ovaa, H, Von Delft, F, London, N
Published 2019Journal article