Novel Histone Deacetylase (HDAC) Inhibitor Induces Apoptosis and Suppresses Invasion via E-Cadherin Upregulation in Pancreatic Ductal Adenocarcinoma (PDAC) by Katja Schiedlauske, Alina Deipenbrock, Marc Pflieger, Alexandra Hamacher, Jan Hänsel, Matthias U. Kassack, Thomas Kurz, Nicole E. Teusch

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The Diverse Binding Modes Explain the Nanomolar Levels of Inhibitory Activities Against 1-Deoxy-<span style="font-variant: small-caps">d</span>-Xylulose 5-Phosphate Reductoisomeras... by Sana Takada, Mona A. Abdullaziz, Stefan Höfmann, Talea Knak, Shin-ichiro Ozawa, Yasumitsu Sakamoto, Thomas Kurz, Nobutada Tanaka

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Over 40 Years of Fosmidomycin Drug Research: A Comprehensive Review and Future Opportunities by Talea Knak, Mona A. Abdullaziz, Stefan Höfmann, Leandro A. Alves Avelar, Saskia Klein, Matthew Martin, Markus Fischer, Nobutada Tanaka, Thomas Kurz

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Assessing the Anthelmintic Candidates BLK127 and HBK4 for Their Efficacy on <i>Haemonchus contortus</i> Adults and Eggs, and Their Hepatotoxicity and Biotransformation by Markéta Zajíčková, Lukáš Prchal, Ivan Vokřál, Linh Thuy Nguyen, Thomas Kurz, Robin Gasser, Klára Bednářová, Magdalena Mičundová, Beate Lungerich, Oliver Michel, Lenka Skálová

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Multioctave high-dynamic range optical spectrometer for single-pulse, longitudinal characterization of ultrashort electron bunches by Omid Zarini, Jurjen Couperus Cabadağ, Yen-Yu Chang, Alexander Köhler, Thomas Kurz, Susanne Schöbel, Wolfgang Seidel, Michael Bussmann, Ulrich Schramm, Arie Irman, Alexander Debus

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Development and reliability of the histological THROMBEX-classification rule for thrombotic emboli of acute ischemic stroke patients by Julika Ribbat-Idel, Florian Stellmacher, Florian Jann, Nicolas Kalms, Inke R. König, Marcus Ohlrich, Georg Royl, Stefan Klotz, Thomas Kurz, Andrè Kemmling, Florian C. Roessler

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Phenotypic screening of the ‘Kurz-box’ of chemicals identifies two compounds (BLK127 and HBK4) with anthelmintic activity in vitro against parasitic larval stages of Haemonchus con... by Linh Thuy Nguyen, Thomas Kurz, Sarah Preston, Hjoerdis Brueckmann, Beate Lungerich, H. M. P. Dilrukshi Herath, Anson V. Koehler, Tao Wang, Lenka Skálová, Abdul Jabbar, Robin B. Gasser

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Class I histone deacetylase inhibitor MS-275 attenuates vasoconstriction and inflammation in angiotensin II-induced hypertension. by Yuhee Ryu, Hae Jin Kee, Simei Sun, Young Mi Seok, Sin Young Choi, Gwi Ran Kim, Seung-Jung Kee, Marc Pflieger, Thomas Kurz, Hyung-Seok Kim, Myung Ho Jeong

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Inhibition of the Yersinia pestis Methylerythritol Phosphate Pathway of Isoprenoid Biosynthesis by α‑Phenyl-Substituted Reverse Fosmidomycin Analogues by Haley S. Ball, Misgina Girma, Mosufa Zainab, Honoria Riley, Christoph T. Behrendt, Claudia Lienau, Sarah Konzuch, Leandro A. A. Avelar, Beate Lungerich, Iswarduth Soojhawon, Schroeder M. Noble, Thomas Kurz, Robin D. Couch

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Three Small Molecule Entities (MPK18, MPK334 and YAK308) with Activity against <i>Haemonchus contortus</i> In Vitro by Aya C. Taki, Abdul Jabbar, Thomas Kurz, Beate Lungerich, Guangxu Ma, Joseph J. Byrne, Marc Pflieger, Yodita Asfaha, Fabian Fischer, Bill C. H. Chang, Brad E. Sleebs, Robin B. Gasser

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Impact of Morphine Treatment With and Without Metoclopramide Coadministration on Myocardial and Microvascular Injury in Acute Myocardial Infarction: Insights From the Randomized Mo... by Thomas Stiermaier, Philipp Schaefer, Roza Meyer‐Saraei, Mohammed Saad, Suzanne de Waha‐Thiele, Janine Pöss, Georg Fuernau, Tobias Graf, Thomas Kurz, Alex Frydrychowicz, Jörg Barkhausen, Steffen Desch, Holger Thiele, Ingo Eitel

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Total Synthesis of the Antimycobacterial Natural Product Chlorflavonin and Analogs via a Late-Stage Ruthenium(II)-Catalyzed <i>ortho</i>-C(sp²)-H-Hydroxylation by Alexander Berger, Talea Knak, Anna-Lene Kiffe-Delf, Korana Mudrovcic, Vinayak Singh, Mathew Njoroge, Bjoern B. Burckhardt, Mohanraj Gopalswamy, Beate Lungerich, Lutz Ackermann, Holger Gohlke, Kelly Chibale, Rainer Kalscheuer, Thomas Kurz

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Effects of novel HDAC inhibitors on urothelial carcinoma cells by Aline Kaletsch, Maria Pinkerneil, Michèle J. Hoffmann, Ananda A. Jaguva Vasudevan, Chenyin Wang, Finn K. Hansen, Constanze Wiek, Helmut Hanenberg, Christoph Gertzen, Holger Gohlke, Matthias U. Kassack, Thomas Kurz, Wolfgang A. Schulz, Günter Niegisch

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Positive allosteric modulation of AMPA receptors via PF4778574 leads to reduced demyelination and clinical disability in experimental models of multiple sclerosis by Mustafa Sindi, Michael Dietrich, Diana Klees, Joel Gruchot, Christina Hecker, John Silbereis, Andrea Issberner, Hans-Peter Hartung, Hans-Peter Hartung, Hans-Peter Hartung, Tobias Ruck, Holger Stark, Thomas Kurz, Patrick Küry, Sven G. Meuth, Philipp Albrecht, Philipp Albrecht

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Regulation of STING activity in DNA sensing by ISG15 modification by Chaohui Lin, Edmund Osei Kuffour, Nina V. Fuchs, Christoph G.W. Gertzen, Jesko Kaiser, Maximilian Hirschenberger, Xiao Tang, Haifeng C. Xu, Oliver Michel, Ronny Tao, Alexandra Haase, Ulrich Martin, Thomas Kurz, Ingo Drexler, Boris Görg, Philipp A. Lang, Tom Luedde, Konstantin M.J. Sparrer, Holger Gohlke, Renate König, Carsten Münk

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Effect of driver charge on wakefield characteristics in a plasma accelerator probed by femtosecond shadowgraphy by Susanne Schöbel, Richard Pausch, Yen-Yu Chang, Sébastien Corde, Jurjen Couperus Cabadağ, Alexander Debus, Hao Ding, Andreas Döpp, F Moritz Foerster, Max Gilljohann, Florian Haberstroh, Thomas Heinemann, Bernhard Hidding, Stefan Karsch, Alexander Köhler, Olena Kononenko, Thomas Kurz, Alastair Nutter, Klaus Steiniger, Patrick Ufer, Alberto Martinez de la Ossa, Ulrich Schramm, Arie Irman

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Progress in Hybrid Plasma Wakefield Acceleration by Bernhard Hidding, Ralph Assmann, Michael Bussmann, David Campbell, Yen-Yu Chang, Sébastien Corde, Jurjen Couperus Cabadağ, Alexander Debus, Andreas Döpp, Max Gilljohann, J. Götzfried, F. Moritz Foerster, Florian Haberstroh, Fahim Habib, Thomas Heinemann, Dominik Hollatz, Arie Irman, Malte Kaluza, Stefan Karsch, Olena Kononenko, Alexander Knetsch, Thomas Kurz, Stephan Kuschel, Alexander Köhler, Alberto Martinez de la Ossa, Alastair Nutter, Richard Pausch, Gaurav Raj, Ulrich Schramm, Susanne Schöbel, Andreas Seidel, Klaus Steiniger, Patrick Ufer, Mark Yeung, Omid Zarini, Matt Zepf

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Tacedinaline (CI-994), a class I HDAC inhibitor, targets intrinsic tumor growth and leptomeningeal dissemination in MYC-driven medulloblastoma while making them susceptible to anti... by Arndt Borkhardt, Nan Qin, Stephen T Keir, Darell D Bigner, Allison Cole, Matthias Wölfl, Viktoria Marquardt, Johanna Theruvath, David Pauck, Daniel Picard, Lena Blümel, Mara Maue, Jasmin Bartl, Ulvi Ahmadov, Maike Langini, Frauke-Dorothee Meyer, Joselyn Cruz-Cruz, Claus M Graef, Till Milde, Olaf Witt, Anat Erdreich-Epstein, Gabriel Leprivier, Ulf Kahlert, Anja Stefanski, Kai Stühler, Julia Hauer, Thomas Beez, Christiane B Knobbe-Thomsen, Ute Fischer, Jörg Felsberg, Finn K Hansen, Rajeev Vibhakar, Sujatha Venkatraman, Samuel H Cheshier, Guido Reifenberger, Thomas Kurz, Marc Remke, Siddhartha Mitra

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