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Bicyclic boronate VNRX-5133 inhibits metallo- and serine-β-lactamases by Krajnc, A, Brem, J, Hinchliffe, P, Calvopiña, K, Panduwawala, TD, Lang, PA, Kamps, JJAG, Tyrrell, JM, Widlake, E, Saward, BG, Walsh, TR, Spencer, J, Schofield, CJ
Published 2019Journal article -
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Imitation of β-lactam binding enables broad-spectrum metallo-β-lactamase inhibitors by Brem, J, Panduwawala, T, Hansen, JU, Hewitt, J, Liepins, E, Donets, P, Espina, L, Farley, AJM, Shubin, K, Campillos, GG, Kiuru, P, Shishodia, S, Krahn, D, Leśniak, RK, Schmidt Adrian, J, Calvopiña, K, Turrientes, M-C, Kavanagh, ME, Lubriks, D, Hinchliffe, P, Langley, GW, Aboklaish, AF, Eneroth, A, Backlund, M, Baran, AG, Nielsen, EI, Speake, M, Kuka, J, Robinson, J, Grinberga, S, Robinson, L, McDonough, MA, Rydzik, AM, Leissing, TM, Jimenez-Castellanos, JC, Avison, MB, Da Silva Pinto, S, Pannifer, AD, Martjuga, M, Widlake, E, Priede, M, Hopkins Navratilova, I, Gniadkowski, M, Belfrage, AK, Brandt, P, Yli-Kauhaluoma, J, Bacque, E, Page, MGP, Björkling, F, Tyrrell, JM, Spencer, J, Lang, PA, Baranczewski, P, Cantón, R, McElroy, SP, Jones, PS, Baquero, F, Suna , E, Morrison, A, Walsh, TR, Schofield, CJ
Published 2021Journal article