Showing 1 - 17 results of 17 for search 'Vedadi, M', query time: 0.54s
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Crystal structure and biophysical characterization of human GDP-D-mannose 4, 6-dehydratase by Vedadi, M, Walker, JR, Sharma, S, Houston, SA, Wasney, G, Loppnau, P, Oppermann, U
Published 2004Conference item -
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A scintillation proximity assay for histone demethylases. by Yu, W, Eram, MS, Hajian, T, Szykowska, A, Burgess-Brown, N, Vedadi, M, Brown, P
Published 2014Journal article -
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Bromo-deaza-SAH: a potent and selective DOT1L inhibitor. by Yu, W, Smil, D, Li, F, Tempel, W, Fedorov, O, Nguyen, K, Bolshan, Y, Al-Awar, R, Knapp, S, Arrowsmith, C, Vedadi, M, Brown, P, Schapira, M
Published 2013Journal article -
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Bromo-deaza-SAH: A potent and selective DOT1L inhibitor by Yu, W, Smil, D, Li, F, Tempel, W, Fedorov, O, Nguyen, K, Bolshan, Y, Al-Awar, R, Knapp, S, Arrowsmith, C, Vedadi, M, Brown, P, Schapira, M
Published 2013Journal article -
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SDR goes SGC: A structural genomics initiative by Oppermann, U, Kavanagh, K, Guo, K, Ng, S, Lukacik, P, Wu, X, Dubinina, E, Shafqat, N, Bray, J, Marsden, B, Sharma, S, Vedadi, M, von Delft, F, Sundstrom, M
Published 2006Conference item -
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Inhibition of the SUV4-20 H1 histone methyltransferase increases frataxin expression in Friedreich's ataxia patient cells by Vilema Enriquez, MG, Quinlan, R, Kilfeather, P, Mazzone, R, Saqlain, S, Del Molino Del Barrio, I, Donato, A, Corda, G, Li, F, Vedadi, M, Németh, AH, Brennan, PE, Wade-Martins, R
Published 2020Journal article -
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Chemical screening methods to identify ligands that promote protein stability, protein crystallization, and structure determination. by Vedadi, M, Niesen, F, Allali-Hassani, A, Fedorov, O, Finerty, P, Wasney, G, Yeung, R, Arrowsmith, C, Ball, L, Berglund, H, Hui, R, Marsden, B, Nordlund, P, Sundstrom, M, Weigelt, J, Edwards, A
Published 2006Journal article -
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Discovery of a highly selective cell‐active inhibitor of the histone lysine demethylases KDM2/7 by Gerken, P, Wolstenhume, J, Tumbler, A, Hatch, S, Zhang, Y, Muller, S, Chandler, S, Mair, B, Li, F, Nijman, S, Konietzny, R, Szommer, T, Yapp, C, Fedorov, O, Benesch, J, Vedadi, M, Kessler, B, Kawamura, A, Brennan, P, Smith, M
Published 2017Journal article -
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A chemical toolbox for the study of bromodomains and epigenetic signaling by Wu, Q, Heidenreich, D, Zhou, S, Ackloo, S, Krämer, A, Nakka, K, Lima-Fernandes, E, Deblois, G, Duan, S, Vellanki, R, Li, F, Vedadi, M, Dilworth, J, Lupien, M, Brennan, P, Arrowsmith, C, Müller, S, Fedorov, O, Filippakopoulos, P, Knapp, S
Published 2019Journal article -
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Discovery of a highly selective cell-active inhibitor of the histone lysine demethylases KDM2/7 by Gerken, PA, Wolstenhulme, JR, Tumber, AM, Hatch, SB, Zhang, Y, Müller, S, Chandler, SA, Mair, B, Li, F, Nijman, SMB, Konietzny, R, Szommer, T, Yapp, C, Fedorov, O, Benesch, JLP, Vedadi, M, Kessler, BM, Kawamura, A, Brennan, PE, Smith, MD
Published 2017Journal article -
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Discovery of a potent and selective fragment-like inhibitor of methyllysine reader protein spindlin 1 (SPIN1) by Xiong, Y, Greschik, H, Johansson, C, Seifert, L, Bacher, J, Park, K, Babault, N, Martini, M, Fagan, V, Li, F, Chau, I, Christott, T, Dilworth, D, Barsyte-Lovejoy, D, Vedadi, M, Arrowsmith, C, Brennan, P, Fedorov, O, Jung, M, Farnie, G, Liu, J, Oppermann, U, Schüle, R, Jin, J
Published 2019Journal article -
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A chemical biology toolbox to study protein methyltransferases and epigenetic signaling by Scheer, S, Ackloo, S, Medina, T, Schapira, M, Li, F, Ward, J, Lewis, A, Northrop, J, Richardson, P, Kaniskan, H, Shen, Y, Liu, J, Smil, D, McLeod, D, Zepeda-Velazquez, C, Luo, M, Jin, J, Barsyte-Lovejoy, D, Huber, K, De Carvalho, D, Vedadi, M, Zaph, C, Brown, P, Arrowsmith, C
Published 2019Journal article -
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The Cryptosporidium parvum kinome. by Artz, J, Wernimont, A, Allali-Hassani, A, Zhao, Y, Amani, M, Lin, Y, Senisterra, G, Wasney, G, Fedorov, O, King, O, Roos, A, Lunin, V, Qiu, W, Finerty, P, Hutchinson, A, Chau, I, von Delft, F, MacKenzie, F, Lew, J, Kozieradzki, I, Vedadi, M, Schapira, M, Zhang, C, Shokat, K, Heightman, T, Hui, R
Published 2011Journal article -
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A chemical probe for Tudor domain protein spindlin1 to investigate chromatin function by Fagan, V, Johansson, C, Gileadi, C, Monteiro, O, Dunford, J, Nibhani, R, Philpott, M, Malzahn, J, Wells, G, Farham, R, Cribbs, A, Halidi, N, Li, F, Chau, I, Greschik, H, Velupillai, S, Allali-Hassani, A, Bennett, J, Christott, T, Giroud, C, Lewis, A, Huber, K, Athanasou, N, Bountra, C, Jung, M, Schüle, R, Vedadi, M, Arrowsmith, C, Xiong, Y, Jin, J, Fedorov, O, Farnie, G, Brennan, P, Oppermann, U
Published 2019Journal article -
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Fragment-based discovery of a chemical probe for the PWWP1 domain of NSD3 by Böttcher, J, Dilworth, D, Reiser, U, Neumüller, R, Schleicher, M, Petronczki, M, Zeeb, M, Mischerikow, N, Allali-Hassani, A, Szewczyk, M, Li, F, Kennedy, S, Vedadi, M, Barsyte-Lovejoy, D, Brown, P, Huber, K, Rogers, C, Wells, C, Fedorov, O, Rumpel, K, Zoephel, A, Mayer, M, Wunberg, T, Böse, D, Zahn, S, Arnhof, H, Berger, H, Reiser, C, Hörmann, A, Krammer, T, Corcokovic, M, Sharps, B, Winkler, S, Häring, D, Cockcroft, X, Fuchs, J, Müllauer, B, Weiss-Puxbaum, A, Gerstberger, T, Boehmelt, G, Vakoc, C, Arrowsmith, C, Pearson, M, McConnell, D
Published 2019Journal article