An Intellectual Disability-Related Missense Mutation in Rac1 Prevents LTP Induction by Chen Tian, Yuni Kay, Anastasiia Sadybekov, Anastasiia Sadybekov, Sadhna Rao, Vsevolod Katritch, Vsevolod Katritch, Vsevolod Katritch, Bruce E. Herring, Bruce E. Herring

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It all clicks together: In silico drug discovery becoming mainstream by Antonina L. Nazarova, Vsevolod Katritch

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An autism spectrum disorder-related de novo mutation hotspot discovered in the GEF1 domain of Trio by Anastasiia Sadybekov, Chen Tian, Cosimo Arnesano, Vsevolod Katritch, Bruce E. Herring

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Structural insight into the activation of a class B G-protein-coupled receptor by peptide hormones in live human cells by Lisa Seidel, Barbara Zarzycka, Saheem A Zaidi, Vsevolod Katritch, Irene Coin

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Detection of autism spectrum disorder-related pathogenic trio variants by a novel structure-based approach by Sadhna Rao, Anastasiia Sadybekov, David C. DeWitt, Joanna Lipka, Vsevolod Katritch, Bruce E. Herring

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High resolution structure of the ba3 cytochrome c oxidase from Thermus thermophilus in a lipidic environment. by Theresa Tiefenbrunn, Wei Liu, Ying Chen, Vsevolod Katritch, C David Stout, James A Fee, Vadim Cherezov

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Computational design of thermostabilizing point mutations for G protein-coupled receptors by Petr Popov, Yao Peng, Ling Shen, Raymond C Stevens, Vadim Cherezov, Zhi-Jie Liu, Vsevolod Katritch

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Dynamic Strategic Bond Analysis Yields a Ten-Step Synthesis of 20-nor-Salvinorin A, a Potent κ‑OR Agonist by Jeremy J. Roach, Yusuke Sasano, Cullen L. Schmid, Saheem Zaidi, Vsevolod Katritch, Raymond C. Stevens, Laura M. Bohn, Ryan A. Shenvi

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Structural details of a Class B GPCR-arrestin complex revealed by genetically encoded crosslinkers in living cells by Yasmin Aydin, Thore Böttke, Jordy Homing Lam, Stefan Ernicke, Anna Fortmann, Maik Tretbar, Barbara Zarzycka, Vsevolod V. Gurevich, Vsevolod Katritch, Irene Coin

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Structure-based discovery of potent and selective melatonin receptor agonists by Nilkanth Patel, Xi Ping Huang, Jessica M Grandner, Linda C Johansson, Benjamin Stauch, John D McCorvy, Yongfeng Liu, Bryan Roth, Vsevolod Katritch

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Structure-Based Virtual Screening of Ultra-Large Library Yields Potent Antagonists for a Lipid GPCR by Arman A. Sadybekov, Rebecca L. Brouillette, Egor Marin, Anastasiia V. Sadybekov, Aleksandra Luginina, Anastasiia Gusach, Alexey Mishin, Élie Besserer-Offroy, Jean-Michel Longpré, Valentin Borshchevskiy, Vadim Cherezov, Philippe Sarret, Vsevolod Katritch

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Structural insights on ligand recognition at the human leukotriene B4 receptor 1 by Nairie Michaelian, Anastasiia Sadybekov, Élie Besserer-Offroy, Gye Won Han, Harini Krishnamurthy, Beata A. Zamlynny, Xavier Fradera, Phieng Siliphaivanh, Jeremy Presland, Kerrie B. Spencer, Stephen M. Soisson, Petr Popov, Philippe Sarret, Vsevolod Katritch, Vadim Cherezov

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Molecular mechanism of biased signaling at the kappa opioid receptor by Amal El Daibani, Joseph M. Paggi, Kuglae Kim, Yianni D. Laloudakis, Petr Popov, Sarah M. Bernhard, Brian E. Krumm, Reid H. J. Olsen, Jeffrey Diberto, F. Ivy Carroll, Vsevolod Katritch, Bernhard Wünsch, Ron O. Dror, Tao Che

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In vitro expression and analysis of the 826 human G protein-coupled receptors by Xuechen Lv, Junlin Liu, Qiaoyun Shi, Qiwen Tan, Dong Wu, John J. Skinner, Angela L. Walker, Lixia Zhao, Xiangxiang Gu, Na Chen, Lu Xue, Pei Si, Lu Zhang, Zeshi Wang, Vsevolod Katritch, Zhi-jie Liu, Raymond C. Stevens

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Controlling opioid receptor functional selectivity by targeting distinct subpockets of the orthosteric site by Rajendra Uprety, Tao Che, Saheem A Zaidi, Steven G Grinnell, Balázs R Varga, Abdelfattah Faouzi, Samuel T Slocum, Abdullah Allaoa, András Varadi, Melissa Nelson, Sarah M Bernhard, Elizaveta Kulko, Valerie Le Rouzic, Shainnel O Eans, Chloe A Simons, Amanda Hunkele, Joan Subrath, Ying Xian Pan, Jonathan A Javitch, Jay P McLaughlin, Bryan L Roth, Gavril W Pasternak, Vsevolod Katritch, Susruta Majumdar

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