Pharmacological Profile of KUL-7211, a Selective -Adrenoceptor Agonist, in Isolated Ureteral Smooth Muscle
Since, in the human ureter, both β2- and β3-adrenoceptors mediate adrenergic-stimulation-induced relaxation, selective β2-/β3-adrenoceptor agonists might prove clinically useful for relieving ureteral colic and promoting stone passage. We evaluated the β-adrenoceptor subtype selectivity and ureteral...
Main Authors: | Yoshitaka Tomiyama, Makoto Murakami, Kohichi Hayakawa, Katsuyoshi Akiyama, Yoshinobu Yamazaki, Masami Kojima, Nobuo Shibata, Masuo Akahane |
---|---|
Format: | Article |
Language: | English |
Published: |
Elsevier
2003-01-01
|
Series: | Journal of Pharmacological Sciences |
Online Access: | http://www.sciencedirect.com/science/article/pii/S1347861319326404 |
Similar Items
-
Challenges in β-adrenoceptor agonist drug development
by: Jonathan R. S. Arch
Published: (2011-04-01) -
Effect of α1D-adrenoceptor blocker for the reduction of ureteral contractions
by: Seong Hwi Hong, et al.
Published: (2023-01-01) -
On the Site and Mechanism of Action of β-Adrenoceptor Agonists in the Bladder
by: Karl Erik Andersson
Published: (2017-03-01) -
Paradoxical bronchoconstriction caused by β2-adrenoceptor agonists
by: Khadija Ayed, et al.
Published: (2020-10-01) -
Effect of beta 2-adrenoceptor agonists on serotonin biochemistry and function.
by: Green, A, et al.
Published: (1984)