An Efficient Synthetic Approach Towards Benzo[<i>b</i>]pyrano[2,3-<i>e</i>][1,4]diazepines, and Their Cytotoxic Activity

An Efficient Synthetic Approach Towards Benzo[<i>b</i>]pyrano[2,3-<i>e</i>][1,4]diazepines, and Their Cytotoxic Activity

In search of unprecedented tri and/or tetrapod pharmacophoric conjugates, a series of 32 new 4-ethyl-1<i>H</i>-benzo[<i>b</i>][1,4]diazepin-2(3<i>H</i>)-ones were synthesized and properly elucidated using MS, IR, NMR, and elemental analysis. <i>In vitro</...

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Bibliographic Details
Main Authors:	Islam H. El Azab, Nadia A.A. Elkanzi
Format:	Article
Language:	English
Published:	MDPI AG 2020-04-01
Series:	Molecules
Subjects:	cyclocondensation reaction benzodiazepine <i>N</i>-heterocycles cytotoxic activity
Online Access:	https://www.mdpi.com/1420-3049/25/9/2051

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