Development of a Rapid In Vitro Screening Assay Using Metabolic Inhibitors to Detect Highly Selective Anticancer Agents

Development of a Rapid In Vitro Screening Assay Using Metabolic Inhibitors to Detect Highly Selective Anticancer Agents

Bibliographic Details
Main Authors:	Felagot A. Abebe, Megan D. Hopkins, Suraj N. Vodnala, Robert J. Sheaff, Angus A. Lamar
Format:	Article
Language:	English
Published:	American Chemical Society 2021-07-01
Series:	ACS Omega
Online Access:	https://doi.org/10.1021/acsomega.1c02203

Similar Items

Anticancer drug screening: standardization of in vitro wound healing assay
by: Vitor M. Almeida, et al.
Published: (2020-03-01)

Anticancer drug screening of natural products: In vitro cytotoxicity assays, techniques, and challenges
by: Agustina Setiawati, et al.
Published: (2022-01-01)

1-Benzamido-1,4-dihydropyridine derivatives as anticancer agents: in vitro and in vivo assays
by: Sandra Ardevines, et al.
Published: (2023-02-01)

Discovery of New Glucose Uptake Inhibitors as Potential Anticancer Agents by Non-Radioactive Cell-Based Assays
by: Hsueh-Chih Hung, et al.
Published: (2022-11-01)

Histone deacetylase inhibitors (HDACIs): multitargeted anticancer agents
by: Ververis K, et al.
Published: (2013-02-01)

SGLT2 Inhibitors as Potential Anticancer Agents
by: Debasish Basak, et al.
Published: (2023-06-01)

The Comparison of MTT and CVS Assays for the Assessment of Anticancer Agent Interactions.
by: Lidia Śliwka, et al.
Published: (2016-01-01)

In Silico Identification and In Vitro Evaluation of New ABCG2 Transporter Inhibitors as Potential Anticancer Agents
by: Simone Di Micco, et al.
Published: (2022-12-01)

Non-peptidic cruzain inhibitors with trypanocidal activity discovered by virtual screening and in vitro assay.
by: Helton J Wiggers, et al.
Published: (2013-01-01)

A rapid in vitro assay for evaluating the effects of acetylcholinesterase inhibitors and reactivators in the rat basolateral amygdala
by: Jeffrey S. Thinschmidt, et al.
Published: (2022-11-01)

Multi-Target Chemometric Modelling, Fragment Analysis and Virtual Screening with ERK Inhibitors as Potential Anticancer Agents
by: Amit Kumar Halder, et al.
Published: (2019-10-01)

Recent progress in DNA methyltransferase inhibitors as anticancer agents
by: Zhixiong Zhang, et al.
Published: (2022-12-01)

Development of novel nuclease inhibitors as potential anticancer agents
by: Bielinski, M
Published: (2022)

Synthesis, Anticancer Screening of Some Novel Trimethoxy Quinazolines and VEGFR2, EGFR Tyrosine Kinase Inhibitors Assay; Molecular Docking Studies
by: Abdulmalik S. Altamimi, et al.
Published: (2021-05-01)

In silico assay development for screening of tetracyclic triterpenoids as anticancer agents against human breast cancer cell line MCF7.
by: Om Prakash, et al.
Published: (2014-01-01)

MEDI 16-Inhibitors of the FBP-FUSE interaction as potential anticancer agents
by: Wyrembak, P, et al.
Published: (2007)

Some anticancer agents as effective glutathione S-transferase (GST) inhibitors
by: Gökçe Başak
Published: (2023-11-01)

Rhamnolipid Biosurfactants—Possible Natural Anticancer Agents and Autophagy Inhibitors
by: Severina Semkova, et al.
Published: (2021-06-01)

An Update on Synthesis of Coumarin Sulfonamides as Enzyme Inhibitors and Anticancer Agents
by: Laila Rubab, et al.
Published: (2022-02-01)

In Vitro Anticancer Activity Screening of Novel Fused Thiophene Derivatives as VEGFR-2/AKT Dual Inhibitors and Apoptosis Inducers
by: Rana M. Abdelnaby, et al.
Published: (2022-06-01)

Small-Molecule RAS Inhibitors as Anticancer Agents: Discovery, Development, and Mechanistic Studies
by: Shaila A. Shetu, et al.
Published: (2022-03-01)

In Vitro and In Silico Studies of Quercetin and Daidzin as Selective Anticancer Agents
by: Muhammad Sulaiman Zubair, et al.
Published: (2021-03-01)

Pyridine-Ureas as Potential Anticancer Agents: Synthesis and In Vitro Biological Evaluation
by: Mohamed El-Naggar, et al.
Published: (2018-06-01)

Molecular modelling studies for 4-oxo-1,4-dihydroquinoline-3-carboxamide derivatives as anticancer agents
by: Suraj S. Kapale, et al.
Published: (2019-06-01)

An anticancer agent
by: Othman, Fauziah, et al.
Published: (2009)

Benzothiazole and Chromone Derivatives as Potential ATR Kinase Inhibitors and Anticancer Agents
by: Mykhaylo Frasinyuk, et al.
Published: (2022-07-01)

Synthesis and Biological Evaluation of New Glycoconjugated LDH Inhibitors as Anticancer Agents
by: Felicia D’Andrea, et al.
Published: (2019-09-01)

Histone Deacetylase Inhibitors in Clinical Studies as Templates for New Anticancer Agents
by: Madhusoodanan Mottamal, et al.
Published: (2015-03-01)

Hybrid topoisomerase I and HDAC inhibitors as dual action anticancer agents.
by: Raffaella Cincinelli, et al.
Published: (2018-01-01)

Metal Complexes as DNA Synthesis and/or Repair Inhibitors: Anticancer and Antimicrobial Agents
by: Mpho Phehello Ngoepe, et al.
Published: (2021-12-01)

In silico drug discovery of SIRT2 inhibitors from natural source as anticancer agents
by: Mahmoud A. A. Ibrahim, et al.
Published: (2023-02-01)

Furo[2,3-d]pyrimidine based derivatives as kinase inhibitors and anticancer agents
by: Marwa A. Aziz, et al.
Published: (2016-06-01)

Screening of Health-Associated Oral Bacteria for Anticancer Properties in vitro
by: Divyashri Baraniya, et al.
Published: (2020-10-01)

Comparison of in vitro anticancer drus screening data generated with a tetrazolium assay versus a protein assay against a diverse panel of human tumor cell lines /
by: 411009 Rubinstein, L. V

Anticancer Inhibitors
by: Alessandra Ammazzalorso, et al.
Published: (2022-07-01)

Thieno[2,3-d]pyrimidine based derivatives as kinase inhibitors and anticancer agents
by: Eman Z. Elrazaz, et al.
Published: (2015-12-01)

Purification and Cytotoxicity Assay of TOmato (Lycopersicum esculentum) Leaves Methanol Extract as Potential Anticancer Agent
by: Wan Chik, Wan Dalila, et al.
Published: (2010)

In-vitro and in-vivo studies on plants and the products for possible source of anticancer agents.
by: Rahmat, Asmah
Published: (2001)

Novel Lycorine Derivatives as Anticancer Agents: Synthesis and In Vitro Biological Evaluation
by: Peng Wang, et al.
Published: (2014-02-01)

In vitro Mechanistic Exploration of Novel Spiropyrrolidine Heterocyclic Hybrids as Anticancer Agents
by: Raju Suresh Kumar, et al.
Published: (2020-06-01)