Probe Cocktail to Assess Transporter Function in Sandwich-Cultured Human Hepatocytes

PURPOSE: Probe substrates are used routinely to assess transporter function in vitro. Administration of multiple probe substrates together as a “cocktail” in sandwich-cultured human hepatocytes (SCHH) could increase the throughput of transporter function assessment in a physiologically-relevant in v...

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Bibliographic Details
Main Authors: Cen Guo, Kenneth R. Brouwer, Paul W Stewart, Caroline Mosley, Kim L.R. Brouwer
Format: Article
Language:English
Published: Frontiers Media S.A. 2019-11-01
Series:Journal of Pharmacy & Pharmaceutical Sciences
Online Access:https://journals.library.ualberta.ca/jpps/index.php/JPPS/article/view/30706