Theranostic Value of Multimers: Lessons Learned from Trimerization of Neurotensin Receptor Ligands and Other Targeting Vectors

Theranostic Value of Multimers: Lessons Learned from Trimerization of Neurotensin Receptor Ligands and Other Targeting Vectors

Neurotensin receptor 1 (NTS1) is overexpressed on a variety of cancer entities; for example, prostate cancer, ductal pancreatic adenocarcinoma, and breast cancer. Therefore, it represents an interesting target for the diagnosis of these cancers types by positron emission tomography (PET) [...]

Bibliographic Details
Main Authors:	Simone Maschauer, Jürgen Einsiedel, Dominik Reich, Harald Hübner, Peter Gmeiner, Hans-Jürgen Wester, Olaf Prante, Johannes Notni
Format:	Article
Language:	English
Published:	MDPI AG 2017-03-01
Series:	Pharmaceuticals
Subjects:	neurotensin neurotensin receptor NTS1 positron emission tomography PET gallium68 TRAP multimerization
Online Access:	http://www.mdpi.com/1424-8247/10/1/29

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