Dopamine transporter interaction with blockers and transportable substrates: insights from kinetics study
Competition kinetic analysis was performed to examine the interaction mechanism of the dopamine transporter with dopamine, (S)-amphetamine, and cocaine, which play a central role in drug abuse phenomena connected with the dopaminergic system. Efficient dopamine transporter inhibitor [3H]PE2I was use...
Main Author: | Vladimir Stepanov |
---|---|
Format: | Article |
Language: | English |
Published: |
Estonian Academy Publishers
2023-11-01
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Series: | Proceedings of the Estonian Academy of Sciences |
Subjects: | |
Online Access: | https://kirj.ee/wp-content/plugins/kirj/pub/proc-4-2023-418-425_20231116210913.pdf |
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