Macrocyclic Peptides Uncover a Novel Binding Mode for Reversible Inhibitors of LSD1
| Main Authors: | , , , , , , , , , , , |
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| Format: | Article |
| Language: | English |
| Published: |
American Chemical Society
2020-02-01
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| Series: | ACS Omega |
| Online Access: | https://doi.org/10.1021/acsomega.9b03493 |
| _version_ | 1819126825636331520 |
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| author | Jie Yang Vladimir O. Talibov Stefan Peintner Claire Rhee Vasanthanathan Poongavanam Matthis Geitmann Matteo Rossi Sebastiano Bernd Simon Janosch Hennig Doreen Dobritzsch U. Helena Danielson Jan Kihlberg |
| author_facet | Jie Yang Vladimir O. Talibov Stefan Peintner Claire Rhee Vasanthanathan Poongavanam Matthis Geitmann Matteo Rossi Sebastiano Bernd Simon Janosch Hennig Doreen Dobritzsch U. Helena Danielson Jan Kihlberg |
| author_sort | Jie Yang |
| collection | DOAJ |
| first_indexed | 2024-12-22T08:02:11Z |
| format | Article |
| id | doaj.art-49645015752a4b7e83c6cc6080b839b7 |
| institution | Directory Open Access Journal |
| issn | 2470-1343 |
| language | English |
| last_indexed | 2024-12-22T08:02:11Z |
| publishDate | 2020-02-01 |
| publisher | American Chemical Society |
| record_format | Article |
| series | ACS Omega |
| spelling | doaj.art-49645015752a4b7e83c6cc6080b839b72022-12-21T18:33:13ZengAmerican Chemical SocietyACS Omega2470-13432020-02-01583979399510.1021/acsomega.9b03493Macrocyclic Peptides Uncover a Novel Binding Mode for Reversible Inhibitors of LSD1Jie Yang0Vladimir O. Talibov1Stefan Peintner2Claire Rhee3Vasanthanathan Poongavanam4Matthis Geitmann5Matteo Rossi Sebastiano6Bernd Simon7Janosch Hennig8Doreen Dobritzsch9U. Helena Danielson10Jan Kihlberg11Department of ChemistryBMC, Uppsala University, Uppsala, SwedenDepartment of ChemistryBMC, Uppsala University, Uppsala, SwedenDepartment of ChemistryBMC, Uppsala University, Uppsala, SwedenDepartment of ChemistryBMC, Uppsala University, Uppsala, SwedenDepartment of ChemistryBMC, Uppsala University, Uppsala, SwedenBeactica AB, Uppsala, SwedenDepartment of ChemistryBMC, Uppsala University, Uppsala, SwedenStructural and Computational Biology Unit, EMBL Heidelberg, Heidelberg, GermanyStructural and Computational Biology Unit, EMBL Heidelberg, Heidelberg, GermanyDepartment of ChemistryBMC, Uppsala University, Uppsala, SwedenDepartment of ChemistryBMC, Uppsala University, Uppsala, SwedenDepartment of ChemistryBMC, Uppsala University, Uppsala, Swedenhttps://doi.org/10.1021/acsomega.9b03493 |
| spellingShingle | Jie Yang Vladimir O. Talibov Stefan Peintner Claire Rhee Vasanthanathan Poongavanam Matthis Geitmann Matteo Rossi Sebastiano Bernd Simon Janosch Hennig Doreen Dobritzsch U. Helena Danielson Jan Kihlberg Macrocyclic Peptides Uncover a Novel Binding Mode for Reversible Inhibitors of LSD1 ACS Omega |
| title | Macrocyclic Peptides Uncover a Novel Binding Mode for Reversible Inhibitors of LSD1 |
| title_full | Macrocyclic Peptides Uncover a Novel Binding Mode for Reversible Inhibitors of LSD1 |
| title_fullStr | Macrocyclic Peptides Uncover a Novel Binding Mode for Reversible Inhibitors of LSD1 |
| title_full_unstemmed | Macrocyclic Peptides Uncover a Novel Binding Mode for Reversible Inhibitors of LSD1 |
| title_short | Macrocyclic Peptides Uncover a Novel Binding Mode for Reversible Inhibitors of LSD1 |
| title_sort | macrocyclic peptides uncover a novel binding mode for reversible inhibitors of lsd1 |
| url | https://doi.org/10.1021/acsomega.9b03493 |
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