Mechanism of antagonist ligand binding to REV-ERBα

Mechanism of antagonist ligand binding to REV-ERBα

Abstract REV-ERBα, a therapeutically promising nuclear hormone receptor, plays a crucial role in regulating various physiological processes such as the circadian clock, inflammation, and metabolism. However, the availability of chemical probes to investigate the pharmacology of this receptor is limi...

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Bibliographic Details
Main Authors:	Mohammad Homaidur Rahman, Lamees Hegazy
Format:	Article
Language:	English
Published:	Nature Portfolio 2024-04-01
Series:	Scientific Reports
Online Access:	https://doi.org/10.1038/s41598-024-58945-4

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