Enantioselective Synthesis of (R)‑Sitagliptin via Phase-Transfer Catalytic aza-Michael Addition

Bibliographic Details
Main Authors: Daehyun Oh, Jaeyong Lee, Sehun Yang, So Hyun Jung, Mihyun Kim, Geumwoo Lee, Hyeung-geun Park
Format: Article
Language:English
Published: American Chemical Society 2024-03-01
Series:ACS Omega
Online Access:https://doi.org/10.1021/acsomega.3c10080
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author Daehyun Oh
Jaeyong Lee
Sehun Yang
So Hyun Jung
Mihyun Kim
Geumwoo Lee
Hyeung-geun Park
author_facet Daehyun Oh
Jaeyong Lee
Sehun Yang
So Hyun Jung
Mihyun Kim
Geumwoo Lee
Hyeung-geun Park
author_sort Daehyun Oh
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spelling doaj.art-4f17bf4f10cd40b5ad14e77a7ee8f33d2024-04-02T08:44:22ZengAmerican Chemical SocietyACS Omega2470-13432024-03-01913153281533810.1021/acsomega.3c10080Enantioselective Synthesis of (R)‑Sitagliptin via Phase-Transfer Catalytic aza-Michael AdditionDaehyun Oh0Jaeyong Lee1Sehun Yang2So Hyun Jung3Mihyun Kim4Geumwoo Lee5Hyeung-geun Park6Research Institute of Pharmaceutical Sciences and College of Pharmacy, Seoul National University, Seoul, Republic of KoreaResearch Institute of Pharmaceutical Sciences and College of Pharmacy, Seoul National University, Seoul, Republic of KoreaResearch Institute of Pharmaceutical Sciences and College of Pharmacy, Seoul National University, Seoul, Republic of KoreaResearch Institute of Pharmaceutical Sciences and College of Pharmacy, Seoul National University, Seoul, Republic of KoreaCollege of Pharmacy, Gachon University, Incheon, Republic of KoreaResearch Institute of Pharmaceutical Sciences and College of Pharmacy, Seoul National University, Seoul, Republic of KoreaResearch Institute of Pharmaceutical Sciences and College of Pharmacy, Seoul National University, Seoul, Republic of Koreahttps://doi.org/10.1021/acsomega.3c10080
spellingShingle Daehyun Oh
Jaeyong Lee
Sehun Yang
So Hyun Jung
Mihyun Kim
Geumwoo Lee
Hyeung-geun Park
Enantioselective Synthesis of (R)‑Sitagliptin via Phase-Transfer Catalytic aza-Michael Addition
ACS Omega
title Enantioselective Synthesis of (R)‑Sitagliptin via Phase-Transfer Catalytic aza-Michael Addition
title_full Enantioselective Synthesis of (R)‑Sitagliptin via Phase-Transfer Catalytic aza-Michael Addition
title_fullStr Enantioselective Synthesis of (R)‑Sitagliptin via Phase-Transfer Catalytic aza-Michael Addition
title_full_unstemmed Enantioselective Synthesis of (R)‑Sitagliptin via Phase-Transfer Catalytic aza-Michael Addition
title_short Enantioselective Synthesis of (R)‑Sitagliptin via Phase-Transfer Catalytic aza-Michael Addition
title_sort enantioselective synthesis of r sitagliptin via phase transfer catalytic aza michael addition
url https://doi.org/10.1021/acsomega.3c10080
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