<i>rel</i>-2-[4-Chloro-2-[(5<i>R</i>,6<i>R</i>,7<i>S</i>)-6-[5-(4-methoxyphenyl)-3-(2-naphthyl)-3,4-dihydropyrazole-2-carbonyl]-5-methyl-2-oxo-3,5,6,7-tetrahydrothiopyrano[2,3-<i>d</i>]thiazol-7-yl]phenoxy]acetic Acid

<i>rel</i>-2-[4-Chloro-2-[(5<i>R</i>,6<i>R</i>,7<i>S</i>)-6-[5-(4-methoxyphenyl)-3-(2-naphthyl)-3,4-dihydropyrazole-2-carbonyl]-5-methyl-2-oxo-3,5,6,7-tetrahydrothiopyrano[2,3-<i>d</i>]thiazol-7-yl]phenoxy]acetic Acid

The hetero-Diels–Alder reaction is the main synthetic tool for obtaining pharmacological agents with a thiopyrano[2,3-<i>d</i>]thiazole motif. In the present work, an efficient method for the synthesis of pyrazoline-containing thiopyrano[2,3-<i>d</i>]thiazole is described. Th...

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Bibliographic Details
Main Authors:	Ihor Yushyn, Serhii Holota, Oksana Ivantsiv, Roman Lesyk
Format:	Article
Language:	English
Published:	MDPI AG 2022-07-01
Series:	Molbank
Subjects:	thiopyrano[2,3-<i>d</i>]thiazoles pyrazoline acylation hetero-Diels–Alder reaction
Online Access:	https://www.mdpi.com/1422-8599/2022/3/M1410

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