Evaluation of Thio- and Seleno-Acetamides Bearing Benzenesulfonamide as Inhibitor of Carbonic Anhydrases from Different Pathogenic Bacteria

Evaluation of Thio- and Seleno-Acetamides Bearing Benzenesulfonamide as Inhibitor of Carbonic Anhydrases from Different Pathogenic Bacteria

A series of 2-thio- and 2-seleno-acetamides bearing the benzenesulfonamide moiety were evaluated as Carbonic Anhydrase (CA, EC 4.2.1.1) inhibitors against different pathogenic bacteria such as the <i>Vibrio cholerae</i> (VchCA-α and VchCA-β), <i>Burkholderia pseud...

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Bibliographic Details
Main Authors:	Andrea Angeli, Mariana Pinteala, Stelian S. Maier, Bogdan C. Simionescu, Andrea Milaneschi, Ghulam Abbas, Sonia del Prete, Clemente Capasso, Antonella Capperucci, Damiano Tanini, Fabrizio Carta, Claudiu T. Supuran
Format:	Article
Language:	English
Published:	MDPI AG 2020-01-01
Series:	International Journal of Molecular Sciences
Subjects:	carbonic anhydrase inhibitors metalloenzymes selenium <i>vibrio cholera</i> <i>burkholderia pseudomallei</i> <i>mycobacterium tuberculosis</i> salmonella
Online Access:	https://www.mdpi.com/1422-0067/21/2/598

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