Microwave-Assisted Synthesis and Butyrylcholinesterase Inhibitory Activity of New Azobenzene Derivatives

Microwave-Assisted Synthesis and Butyrylcholinesterase Inhibitory Activity of New Azobenzene Derivatives

Cholinesterase inhibitors (ChEis) play an important role in enhancing cholinergic synaptic activity and, consequently, have therapeutic applications in the treatment of neurodegenerative diseases like Alzheimer’s disease (AD). The inhibition of the enzymes acetylcholinesterase (AChE) and butyrylchol...

Full description

Bibliographic Details
Main Authors:	Martina Donozo, Valeria Cavallaro, Ana Paula Murray, Carlos Javier Baier
Format:	Article
Language:	English
Published:	MDPI AG 2022-11-01
Series:	Medical Sciences Forum
Subjects:	azobenzene Alzheimer’s disease butyrylcholinesterase microwave cytotoxic
Online Access:	https://www.mdpi.com/2673-9992/14/1/31

Similar Items

Microwave Assisted Synthesis of BenzilideneBenzylamine and Its Acetylcholinesterase and Butyrylcholinesterase Activity
by: Himayat Ullah, et al.
Published: (2020-12-01)

Rivastigmine–Bambuterol Hybrids as Selective Butyrylcholinesterase Inhibitors
by: Jie Wu, et al.
Published: (2023-12-01)

Azobenzene as Antimicrobial Molecules
by: Miriam Di Martino, et al.
Published: (2022-09-01)

Identification of a Novel Dual Inhibitor of Acetylcholinesterase and Butyrylcholinesterase: In Vitro and In Silico Studies
by: Raquel B. M. de Almeida, et al.
Published: (2023-01-01)

LIGHT-DRIVEN MOLECULAR MOTORS BASED ON AZOBENZENE PHOTOIZOMERIZATION
by: Rodica-Mariana ION, et al.
Published: (2010-05-01)

Butyrylcholinesterase inhibitory activity of peptides identified from yellow field pea (Pisum sativum) enzymatic protein hydrolysates
by: Nancy D. Asen, et al.
Published: (2023-07-01)

Inhibition of acetylcholinesterase and butyrylcholinesterase with uracil derivatives: kinetic and computational studies
by: Huseyin Cavdar, et al.
Published: (2019-01-01)

Inhibitory Effects of Cannabinoids on Acetylcholinesterase and Butyrylcholinesterase Enzyme Activities
by: Tess Puopolo, et al.
Published: (2022-04-01)

Phlorotannins from Ishige okamurae and their acetyl- and butyrylcholinesterase inhibitory effects
by: Na Young Yoon, et al.
Published: (2009-10-01)

New Resveratrol Derivatives Exhibit Acetylcholinesterase Inhibitory Properties and Decrease Reactive Oxygen Species Production in the SH-SY5Y Human Neuroblastoma Cell Line
by: Martina Donozo, et al.
Published: (2023-03-01)

Evaluation of the Key Structural Features of Various Butyrylcholinesterase Inhibitors Using Simple Molecular Descriptors
by: Ante Miličević, et al.
Published: (2022-10-01)

Azobenzene/Tetraethyl Ammonium Photochromic Potassium Channel Blockers: Scope and Limitations for Design of Para-Substituted Derivatives with Specific Absorption Band Maxima and Thermal Isomerization Rate
by: Daniil M. Strashkov, et al.
Published: (2021-12-01)

Estudos de QSAR 3D para um conjunto de inibidores de butirilcolinesterase humana QSAR 3D studies of a series of human butyrylcholinesterase inhibitors
by: Humberto F. Freitas, et al.
Published: (2009-01-01)

Triterpene-Based Carboxamides Act as Good Inhibitors of Butyrylcholinesterase
by: Anne Loesche, et al.
Published: (2019-03-01)

Fluorescent Azobenzene-Containing Compounds: From Structure to Mechanism
by: Lulu Xue, et al.
Published: (2021-07-01)

Biphenylalkoxyamine Derivatives–Histamine H<sub>3</sub> Receptor Ligands with Butyrylcholinesterase Inhibitory Activity
by: Dorota Łażewska, et al.
Published: (2021-06-01)

Molecular interaction of inhibitors with human brain butyrylcholinesterase
by: Shazi Shakil
Published: (2021-11-01)

Subchronic Oral Exposure to Chlorpyrifos Decreases Butyrylcholinesterase in Wistar Ra
by: Elly Nurus Sakinah, et al.
Published: (2024-03-01)

Azobenzene‐Based Photomechanical Biomaterials
by: Jing Sun, et al.
Published: (2021-09-01)

The Role of Butyrylcholinesterase and Iron in the Regulation of Cholinergic Network and Cognitive Dysfunction in Alzheimer’s Disease Pathogenesis
by: Jacek Jasiecki, et al.
Published: (2021-02-01)

Amino-7,8-dihydro-4H-chromenone derivatives as potential inhibitors of acetylcholinesterase and butyrylcholinesterase for Alzheimer’s disease management; in vitro and in silico study
by: Ali Asadipour, et al.
Published: (2024-04-01)

An azobenzene container showing a definite folding – synthesis and structural investigation
by: Abdulselam Adam, et al.
Published: (2019-07-01)

Evaluation of Acetyl- and Butyrylcholinesterase Enzyme Inhibitory Activities and Cytotoxic Activities of Anthraquinone Derivatives
by: Funda OZKOK, et al.
Published: (2022-08-01)

Synthesis and biological evaluation of lycorine derivatives as dual inhibitors of human acetylcholinesterase and butyrylcholinesterase
by: Wang Yue-Hu, et al.
Published: (2012-09-01)

Machine learning modeling of the absorption properties of azobenzene molecules
by: Valentin Stanev, et al.
Published: (2023-06-01)

Reconfigurable and Recyclable Photoactuators Based on Azobenzene-Containing Polymers
by: Mingsen Chen, et al.
Published: (2020-08-01)

Photodynamic control of bacterial motility by means of azobenzene molecules
by: Ismaël Duchesne, et al.
Published: (2021-12-01)

Novel anti-neuroinflammatory pyranone-carbamate derivatives as selective butyrylcholinesterase inhibitors for treating Alzheimer’s disease
by: Chuanyu Yu, et al.
Published: (2024-12-01)

Synthesis of photoresponsive cholesterol-based azobenzene organogels: dependence on different spacer lengths
by: Yuchun Ren, et al.
Published: (2015-06-01)

Reprocessable Photodeformable Azobenzene Polymers
by: Huiqi Zhang
Published: (2021-07-01)

Evaluation of N-alkyl isatins and indoles as acetylcholinesterase and butyrylcholinesterase inhibitors
by: Kaitlyn N. Alcorn, et al.
Published: (2024-12-01)

Butyrylcholinesterase deficiency identified after succinylcholine administration. Case report
by: Manzano Rincón, Yolima, et al.
Published: (2018-01-01)

Development of potent reversible selective inhibitors of butyrylcholinesterase as fluorescent probes
by: Stane Pajk, et al.
Published: (2020-01-01)

Responsive Azobenzene-Containing Polymers and Gels
by: Deshmukh, Smeet, et al.
Published: (2004)

Redshifting azobenzenes for photoswitchable ion transport and catalysis
by: Kerckhoffs, A
Published: (2023)

Discovery of new butyrylcholinesterase inhibitors via structure-based virtual screening
by: Noor Atatreh, et al.
Published: (2019-01-01)

Discovery of pyrrole derivatives as acetylcholinesterase-sparing butyrylcholinesterase inhibitor
by: Shouyuan Sun, et al.
Published: (2022-12-01)

Pursuing the Complexity of Alzheimer’s Disease: Discovery of Fluoren-9-Amines as Selective Butyrylcholinesterase Inhibitors and <i>N</i>-Methyl-<span style="font-variant: small-caps">d</span>-Aspartate Receptor Antagonists
by: Jan Konecny, et al.
Published: (2020-12-01)

Synthesis and photochromism of catechol-containing symmetrical azobenzene compounds
by: Suju Fan, et al.
Published: (2022-06-01)

Construction of multiresponsive supramacromolecular hydrogels with a novel azobenzene derivative as crosslinkers
by: Tianhao Wang, et al.
Published: (2023-01-01)