Synthesis and Antibacterial Evaluation of New Sulfone Derivatives Containing 2-Aroxymethyl-1,3,4-Oxadiazole/Thiadiazole Moiety

Synthesis and Antibacterial Evaluation of New Sulfone Derivatives Containing 2-Aroxymethyl-1,3,4-Oxadiazole/Thiadiazole Moiety

Sulfones are one of the most important classes of agricultural fungicides. To discover new lead compounds with high antibacterial activity, a series of new sulfone derivatives were designed and synthesized by introducing the aroxymethyl moiety into the scaffold of 1,3,4-oxadiazole/thiadiazole sulfon...

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Bibliographic Details
Main Authors:	Shihu Su, Xia Zhou, Guoping Liao, Puying Qi, Linhong Jin
Format:	Article
Language:	English
Published:	MDPI AG 2016-12-01
Series:	Molecules
Subjects:	synthesis 1,3,4-oxadiazole/thiadiazole sulfone aryloxymethyl antibacterial activity structure-activity relationship
Online Access:	http://www.mdpi.com/1420-3049/22/1/64

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