Amination of 5-Spiro-Substituted 3-Hydroxy-1,5-dihydro-2<i>H</i>-pyrrol-2-ones
The 3-hydroxy-1,5-dihydro-2<i>H</i>-pyrrol-2-one motif is a valuable scaffold in drug discovery. The replacement of the 3-oxy fragment in 3-hydroxy-1,5-dihydro-2<i>H</i>-pyrrol-2-ones-based compounds with a 3-amino one (3-amino analogs of 3-hydroxy-1,5-dihydro-2<i>H<...
Main Authors: | , , , , |
---|---|
Format: | Article |
Language: | English |
Published: |
MDPI AG
2021-11-01
|
Series: | Molecules |
Subjects: | |
Online Access: | https://www.mdpi.com/1420-3049/26/23/7179 |