Pharmacological Profiles of Oligomerized μ-Opioid Receptors

Pharmacological Profiles of Oligomerized μ-Opioid Receptors

Opioids are widely prescribed pain relievers with multiple side effects and potential complications. They produce analgesia via G-protein-protein coupled receptors: μ-, δ-, κ-opioid and opioid receptor-like 1 receptors. Bivalent ligands targeted to the oligomerized opioid receptors might be the key...

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Bibliographic Details
Main Authors:	Ing-Kang Ho, Cynthia Wei-Sheng Lee
Format:	Article
Language:	English
Published:	MDPI AG 2013-10-01
Series:	Cells
Subjects:	μ-opioid receptor bivalent ligand receptor oligomerization
Online Access:	http://www.mdpi.com/2073-4409/2/4/689

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