[1,5]-Hydride Shift-Cyclization <i>versus</i> C(sp<sup>2</sup>)-H Functionalization in the Knoevenagel-Cyclization Domino Reactions of 1,4- and 1,5-Benzoxazepines
Domino cyclization reactions of <i>N</i>-aryl-1,4- and 1,5-benzoxazepine derivatives involving [1,5]-hydride shift or C(sp<sup>2</sup>)-H functionalization were investigated. Neuroprotective and acetylcholinesterase activities of the products were studied. Domino Knoevenagel-...
Main Authors: | Dóra Szalóki Vargáné, László Tóth, Balázs Buglyó, Attila Kiss-Szikszai, Attila Mándi, Péter Mátyus, Sándor Antus, Yinghan Chen, Dehai Li, Lingxue Tao, Haiyan Zhang, Tibor Kurtán |
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Format: | Article |
Language: | English |
Published: |
MDPI AG
2020-03-01
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Series: | Molecules |
Subjects: | |
Online Access: | https://www.mdpi.com/1420-3049/25/6/1265 |
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