Biological Docking and BSA Binding Studies of 1,4-Disubstituted Piperdine Containing 1,2,4-Triazoles: Comparative Synthesis Leveraging Microwave-Assisted and Conventional Protocols

Biological Docking and BSA Binding Studies of 1,4-Disubstituted Piperdine Containing 1,2,4-Triazoles: Comparative Synthesis Leveraging Microwave-Assisted and Conventional Protocols

A biologically effective study regarding the synthesis of a library of hybrids based on a triazole ring, propanamide and azinane was performed in this study. The targeted hybrids, <b>9a–9l</b>, were synthesized through a multistep protocol followed by two methodologies, that is, conventi...

Bibliográfalaš dieđut
Váldodahkkit:	Javed Iqbal, Naeem Akhtar Virk, Aziz Ur Rehman, Aleksey Kuznetsov, Shahid Rasool, Muhammad Yasir, Syed Adnan Ali Shah
Materiálatiipa:	Artihkal
Giella:	English
Almmustuhtton:	MDPI AG 2023-11-01
Ráidu:	Chemistry Proceedings
Fáttát:	triazole azinane enzymes molecular docking BSA binding
Liŋkkat:	https://www.mdpi.com/2673-4583/14/1/106

Geahča maid

Synthesis of some New 1,2,4-Triazole derivatives
Dahkki: Ibtehal Kahtan Abdullah
Almmustuhtton: (2013-11-01)

Thermal Rearrangement of Allyl Substituted Unsymmetric 4H-1,2,4-Triazoles to the Corresponding 1H-1,2,4-triazoles
Dahkki: Per H.J. Carlsen, et al.
Almmustuhtton: (2001-04-01)

Regioselectivity in the Thermal Rearrangement of Unsymmetrical 4-Methyl-4H-1,2,4-triazoles to 1-Methyl-1H-1,2,4-triazoles
Dahkki: Per H.J. Carlsen, et al.
Almmustuhtton: (2001-11-01)

Synthesis Some of New Substituted 1,3,4-Thiadiazole and 1,2,4-Triazole
Dahkki: Tamara alsafar, et al.
Almmustuhtton: (2020-03-01)

Synthesis and biological activities of 3,6-disubstituted-1,2,4-triazolo-1,3,4- thiadiazole derivatives
Dahkki: L. Lin,, et al.
Almmustuhtton: (2018-01-01)

Synthesis methods of 1,2,3-/1,2,4-triazoles: A review
Dahkki: Jinlian Dai, et al.
Almmustuhtton: (2022-09-01)

1,2,4-Triazoles as Important Antibacterial Agents
Dahkki: Małgorzata Strzelecka, et al.
Almmustuhtton: (2021-03-01)

Synthesis and Biological Activities of Some 1,2,4-Triazole Derivatives: A Review
Dahkki: Dina Saleem M. Ameen, et al.
Almmustuhtton: (2022-10-01)

Synthesis of New Bis-1,2,4-Triazole Derivatives
Dahkki: Hakan Bektas, et al.
Almmustuhtton: (2006-06-01)

New 1,2,3-Triazole/1,2,4-triazole Hybrids as Aromatase Inhibitors: Design, Synthesis, and Apoptotic Antiproliferative Activity
Dahkki: Mohamed T-E Maghraby, et al.
Almmustuhtton: (2023-10-01)

Combination of 1,2,3-triazole and 1,2,4-triazole frameworks for new high-energy and low-sensitivity compounds
Dahkki: Wenjing Yao, et al.
Almmustuhtton: (2021-06-01)

Highly Efficient Synthesis of 1,4-Disubstituted 1,2,3-Triazole Derivatives under Ultrasonic Irradiation, Evaluation of Vasorelaxant Activities
Dahkki: Sakineh Ebrahimpourmoghaddam, et al.
Almmustuhtton: (2024-03-01)

Synthesis Of 2-Benzamidomethyl-5-Substituted Amino-1,3,4-Thiadiazoles-2,5-Disubstituted 1,3,4-Oxadiazole and 4,5-Disubstituted 1,2,4-Triazole-3-Thiol
Dahkki: K. M. Daoud, et al.
Almmustuhtton: (2012-12-01)

1-[({5-[(4-Methylphenoxy)methyl]-4-phenyl-4H-1,2,4-triazol-3-yl}sulfanyl)methyl]-1H-benzo[d][1,2,3]triazole
Dahkki: Shaaban K. Mohamed, et al.
Almmustuhtton: (2016-11-01)

Synthesis and crystal structure of 3-(adamantan-1-yl)-4-(2-bromo-4-fluorophenyl)-1H-1,2,4-triazole-5(4H)-thione
Dahkki: Alaa S. Abdelrazeq, et al.
Almmustuhtton: (2020-02-01)

Synthesis and Characterization of the Triazole Derived from Thiosemicarbazide, 4-Amino-5-Phenyl-4H-1,2,4- Triazole-3-Thiol and Their Copper(II) and Nickel(II) Complexes
Dahkki: Hamdan Abood Aday
Almmustuhtton: (2013-02-01)

Corrosion of α-Brass in Solutions Containing Chloride Ions and 3-Mercaptoalkyl-5-amino-1<em>H</em>-1,2,4-triazoles
Dahkki: Oleg Kozaderov, et al.
Almmustuhtton: (2019-07-01)

Synthesis and alkylation of 5-aryl-1,2-dihydro-3H-1,2,4-triazole-3-thiones
Dahkki: Dmytro V. Dovbnya, et al.
Almmustuhtton: (2021-06-01)

Synthesis of some substituted 1,3,4-oxadiazoles, thiadiazoles and 1,2,4-triazoles
Dahkki: Shereen R. Mohamed
Almmustuhtton: (2009-06-01)

5-[(2-Isopropyl-5-methylphenoxy)methyl]-4-phenyl-4H-1,2,4-triazole-3-thiol
Dahkki: Abdullah Mohamed Asiri
Almmustuhtton: (2003-02-01)

Theoretical Study of Tautomeric Conformations for 1,2,4-Triazole Derivatives
Dahkki: Radia Mahboub
Almmustuhtton: (2021-03-01)

The synthesis and study of physicochemical properties of 1,2,4-triazole derivatives containing the phenethyl group in position 5
Dahkki: Tetiana V. Ihnatova, et al.
Almmustuhtton: (2020-05-01)

2-({5-[(4-Chlorophenoxy)methyl]-4-phenyl-4H-1,2,4-triazol-3-yl}sulfanyl)-N-phenylacetamide
Dahkki: Joel T. Mague, et al.
Almmustuhtton: (2016-03-01)

1,3-Bis(1,2,4-triazol-1-yl)adamantane
Dahkki: Roman Marchenko, et al.
Almmustuhtton: (2017-12-01)

3-Ethoxy-5-phenyl-1H-1,2,4-triazole
Dahkki: Ali M. Hebishy, et al.
Almmustuhtton: (2019-04-01)

Synthesis, antimycobacterial evaluation, and molecular docking study of 1,2,4-triazole derivatives
Dahkki: Meng-Yu Xia, et al.
Almmustuhtton: (2023-12-01)

Design, synthesis, and antiproliferative activity of novel 1,2,4-triazole-chalcone compounds
Dahkki: Li Jinjing, et al.
Almmustuhtton: (2023-10-01)

Toxicity prediction of 1,2,4-triazoles compounds by QSTR and interspecies QSTTR models
Dahkki: Zhiyong Liu, et al.
Almmustuhtton: (2022-09-01)

In vitro Biological Evaluation of 1,2,4-triazole Mannich Base
Dahkki: Mahmood Sherzad Rafaat, et al.
Almmustuhtton: (2023-12-01)

Synthesis of 3,5-di-(4-pyridyl)-1H-1,2,4-triazole
Dahkki: Guang Yang, et al.
Almmustuhtton: (2008-03-01)

Synthesis, Characterization and Antifungal Evaluation of 5-Substituted-4-Amino-1,2,4-Triazole-3-Thioesters
Dahkki: Aurangzeb Hasan, et al.
Almmustuhtton: (2011-01-01)

Determination of antimicrobial activity of some 1,2,4-triazole derivatives
Dahkki: M. S. M. Alrawashdeh
Almmustuhtton: (2018-04-01)

Proton-Conducting Polymeric Membranes Based on 1,2,4-Triazole
Dahkki: Galina F. Prozorova, et al.
Almmustuhtton: (2023-01-01)

Synthesis, antibacterial and surface activity of 1,2,4-triazole derivatives
Dahkki: R. El-Sayed
Almmustuhtton: (2006-06-01)

Synthesis of Chiral 1,4-Disubstituted-1,2,3-Triazole Derivatives from Amino Acids
Dahkki: Morten Grøtli, et al.
Almmustuhtton: (2009-12-01)

Synthesis of novel indole, 1,2,4-triazole derivatives as potential glucosidase inhibitors
Dahkki: Ramesh S Gani, et al.
Almmustuhtton: (2020-12-01)

Green ultrasound-assisted three-component click synthesis of novel 1H-1,2,3-triazole carrying benzothiazoles and fluorinated-1,2,4-triazole conjugates and their antimicrobial evaluation
Dahkki: Rezki Nadjet, et al.
Almmustuhtton: (2017-09-01)

Crystal structure of 2-{[5-(methylsulfanyl)-4-phenyl-4H-1,2,4-triazol-3-yl]methyl}benzo[d]thiazole
Dahkki: Rasha A. Azzam, et al.
Almmustuhtton: (2023-09-01)

N-[(E)-Quinolin-2-ylmethylidene]-1,2,4-triazol-4-amine hemihydrate
Dahkki: Nurulizzatul Ningsheh M. Shahri, et al.
Almmustuhtton: (2020-02-01)

Enantiomer stability of atropisomeric 1,5-disubstituted 1,2,3-triazoles
Dahkki: Fernanda Meloni, et al.
Almmustuhtton: (2022-03-01)