Novel anti-neuroinflammatory pyranone-carbamate derivatives as selective butyrylcholinesterase inhibitors for treating Alzheimer’s disease

Butyrylcholinesterase (BuChE) and neuroinflammation have recently emerged as promising therapeutic directions for Alzheimer’s disease (AD). Herein, we synthesised 19 novel pyranone-carbamate derivatives and evaluated their activities against cholinesterases and neuroinflammation. The optimal compoun...

詳細記述

書誌詳細
主要な著者: Chuanyu Yu, Xueyan Liu, Bingxiang Ma, Jiexin Xu, Yiquan Chen, Chaoxian Dai, Huaping Peng, Daijun Zha
フォーマット: 論文
言語:English
出版事項: Taylor & Francis Group 2024-12-01
シリーズ:Journal of Enzyme Inhibition and Medicinal Chemistry
主題:
オンライン・アクセス:https://www.tandfonline.com/doi/10.1080/14756366.2024.2313682