Microwave-Assisted Sequential One-Pot Synthesis of 8-Substituted Pyrazolo[1,5-<i>a</i>][1,3,5]triazines

Microwave-Assisted Sequential One-Pot Synthesis of 8-Substituted Pyrazolo[1,5-<i>a</i>][1,3,5]triazines

This paper reports a convenient sequential one-pot approach for the synthesis of an array of 14 pyrazolo[1,5-<i>a</i>][1,3,5]triazines, substituted in C8 by halogen (Br), various functions (CN and CO<sub>2</sub>Et) and alkyl or (het)aryl groups. This study confirms the intere...

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Bibliographic Details
Main Authors:	Jonathan Elie, Corinne Fruit, Thierry Besson
Format:	Article
Language:	English
Published:	MDPI AG 2021-06-01
Series:	Molecules
Subjects:	microwave-assisted chemistry one-pot synthesis pyrazolo[1,5-<i>a</i>][1,3,5]triazines 5-aza-9-deazapurines
Online Access:	https://www.mdpi.com/1420-3049/26/12/3540

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