An alternative synthesis of Azilsartan: an angiotensin II receptor blocker
This paper provides a description of an alternative, novel and commercially viable process which has been developed for the preparation of Azilsartan, a pro-drug of Azilsartan medoxomil, an angiotensin II receptor blocker. The present work also provides a primary account of the synthesis and charact...
| Main Authors: | , , , , , , |
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| Format: | Article |
| Language: | English |
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Sciendo
2015-06-01
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| Series: | Current Issues in Pharmacy and Medical Sciences |
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| Online Access: | https://doi.org/10.1515/cipms-2015-0047 |
| _version_ | 1818728035885514752 |
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| author | Garaga Srinivas Misra Nimesh C. Reddy Ambati V. Raghava Prabahar Koilpillai Joseph Takshinamoorthy Chandiran Sanasi Paul Douglas Korupolu Raghubabu |
| author_facet | Garaga Srinivas Misra Nimesh C. Reddy Ambati V. Raghava Prabahar Koilpillai Joseph Takshinamoorthy Chandiran Sanasi Paul Douglas Korupolu Raghubabu |
| author_sort | Garaga Srinivas |
| collection | DOAJ |
| description | This paper provides a description of an alternative, novel and commercially viable process which has been developed for the preparation of Azilsartan, a pro-drug of Azilsartan medoxomil, an angiotensin II receptor blocker. The present work also provides a primary account of the synthesis and characterization of the novel intermediates (6, 7 & 10) of Azilsartan, with their spectral data. |
| first_indexed | 2024-12-17T22:23:36Z |
| format | Article |
| id | doaj.art-a5a6b47578fe4dceb2bc9172da4e1482 |
| institution | Directory Open Access Journal |
| issn | 2084-980X 2300-6676 |
| language | English |
| last_indexed | 2024-12-17T22:23:36Z |
| publishDate | 2015-06-01 |
| publisher | Sciendo |
| record_format | Article |
| series | Current Issues in Pharmacy and Medical Sciences |
| spelling | doaj.art-a5a6b47578fe4dceb2bc9172da4e14822022-12-21T21:30:25ZengSciendoCurrent Issues in Pharmacy and Medical Sciences2084-980X2300-66762015-06-01282727610.1515/cipms-2015-0047cipms-2015-0047An alternative synthesis of Azilsartan: an angiotensin II receptor blockerGaraga Srinivas0Misra Nimesh C.1Reddy Ambati V. Raghava2Prabahar Koilpillai Joseph3Takshinamoorthy Chandiran4Sanasi Paul Douglas5Korupolu Raghubabu6Chemical Research and Development Department, Aurobindo Pharma Ltd, Survey No: 71&72, Indrakaran Village, Sangareddy Mandal, Medak district, Hyderabad – 502329, Andhra Pradesh, IndiaChemical Research and Development Department, Aurobindo Pharma Ltd, Survey No: 71&72, Indrakaran Village, Sangareddy Mandal, Medak district, Hyderabad – 502329, Andhra Pradesh, IndiaChemical Research and Development Department, Aurobindo Pharma Ltd, Survey No: 71&72, Indrakaran Village, Sangareddy Mandal, Medak district, Hyderabad – 502329, Andhra Pradesh, IndiaChemical Research and Development Department, Aurobindo Pharma Ltd, Survey No: 71&72, Indrakaran Village, Sangareddy Mandal, Medak district, Hyderabad – 502329, Andhra Pradesh, IndiaChemical Research and Development Department, Aurobindo Pharma Ltd, Survey No: 71&72, Indrakaran Village, Sangareddy Mandal, Medak district, Hyderabad – 502329, Andhra Pradesh, IndiaDepartment of Engineering Chemistry, A. U. College of Engineering (A), Andhra University, Visakhapatnam – 530003, Andhra Pradesh, IndiaDepartment of Engineering Chemistry, A. U. College of Engineering (A), Andhra University, Visakhapatnam – 530003, Andhra Pradesh, IndiaThis paper provides a description of an alternative, novel and commercially viable process which has been developed for the preparation of Azilsartan, a pro-drug of Azilsartan medoxomil, an angiotensin II receptor blocker. The present work also provides a primary account of the synthesis and characterization of the novel intermediates (6, 7 & 10) of Azilsartan, with their spectral data.https://doi.org/10.1515/cipms-2015-0047azilsartannovel intermediatessynthesis and characterization |
| spellingShingle | Garaga Srinivas Misra Nimesh C. Reddy Ambati V. Raghava Prabahar Koilpillai Joseph Takshinamoorthy Chandiran Sanasi Paul Douglas Korupolu Raghubabu An alternative synthesis of Azilsartan: an angiotensin II receptor blocker Current Issues in Pharmacy and Medical Sciences azilsartan novel intermediates synthesis and characterization |
| title | An alternative synthesis of Azilsartan: an angiotensin II receptor blocker |
| title_full | An alternative synthesis of Azilsartan: an angiotensin II receptor blocker |
| title_fullStr | An alternative synthesis of Azilsartan: an angiotensin II receptor blocker |
| title_full_unstemmed | An alternative synthesis of Azilsartan: an angiotensin II receptor blocker |
| title_short | An alternative synthesis of Azilsartan: an angiotensin II receptor blocker |
| title_sort | alternative synthesis of azilsartan an angiotensin ii receptor blocker |
| topic | azilsartan novel intermediates synthesis and characterization |
| url | https://doi.org/10.1515/cipms-2015-0047 |
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