Chemical Strategies towards the Synthesis of Betulinic Acid and Its More Potent Antiprotozoal Analogues

Chemical Strategies towards the Synthesis of Betulinic Acid and Its More Potent Antiprotozoal Analogues

Betulinic acid (BA, 3β-hydroxy-lup-20(29)-en-28-oic acid) is a pentacyclic triterpene acid present predominantly in <i>Betula</i> ssp. (Betulaceae) and is also widely spread in many species belonging to different plant families. BA presents a wide spectrum of remarkable pharmacological p...

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Bibliographic Details
Main Authors:	André Barreto Cunha, Ronan Batista, María Ángeles Castro, Jorge Mauricio David
Format:	Article
Language:	English
Published:	MDPI AG 2021-02-01
Series:	Molecules
Subjects:	betulinic acid antiprotozoal activities triterpene acid derivatives antiplasmodial activity antileishmanial activity antitrypanosomal activity
Online Access:	https://www.mdpi.com/1420-3049/26/4/1081

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