Arylsulfonamido-alkyl-sulfamates act as inhibitors of bovine carbonic anhydrase II

Arylsulfonamido-alkyl-sulfamates act as inhibitors of bovine carbonic anhydrase II

A small library of arylsulfonamido-alkyl sulfamates was prepared by a two-step synthesis from readily available starting materials. The compounds were tested for their ability to inhibit bovine carbonic anhydrase II. Several of them were found as good competitive inhibitors holding Ki values as low...

Bibliografiset tiedot
Päätekijät:	Toni C. Denner, Niels V. Heise, René Csuk
Aineistotyyppi:	Artikkeli
Kieli:	English
Julkaistu:	Elsevier 2024-12-01
Sarja:	European Journal of Medicinal Chemistry Reports
Aiheet:	Sulfamates Carbonic anhydrase II Inhibitor
Linkit:	http://www.sciencedirect.com/science/article/pii/S2772417424000499

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