Synthesis and biochemical evaluation of (R)-5-acyloxymethyl- and (S)-5-acylaminomethyl-3-(1H-pyrrol-1-yl)-2-oxazolidinones as new anti-monoamine oxidase (anti-MAO) agents

Synthesis and biochemical evaluation of (R)-5-acyloxymethyl- and (S)-5-acylaminomethyl-3-(1H-pyrrol-1-yl)-2-oxazolidinones as new anti-monoamine oxidase (anti-MAO) agents

Bibliographic Details
Main Authors:	Antonello Mai, Marino Artico, Sergio Valente, Ilaria Cerbara, Olivia Befani, Paola Turini Laura Dalla Vedova, Enzo Agostinelli
Format:	Article
Language:	English
Published:	Arkat USA, Inc. 2004-01-01
Series:	ARKIVOC
Online Access:	https://www.arkat-usa.org/arkivoc-journal/browse-arkivoc/ark.5550190.0005.504

Similar Items

N-Acyloxymethyl-phthalimides deliver genotoxic formaldehyde to human cells
by: Emms, VL, et al.
Published: (2023)

Enantiopure oxazolidinones as chiral acids in the asymmetric protonation of N-Boc pyrrole derived enolates.
by: Carbery, DR, et al.
Published: (2004)

β-Carboline Alkaloids in Soy Sauce and Inhibition of Monoamine Oxidase (MAO)
by: Tomás Herraiz
Published: (2023-03-01)

Monoamine Oxidase (MAO) as a Potential Target for Anticancer Drug Design and Development
by: Reem Aljanabi, et al.
Published: (2021-10-01)

Modification, Characterization of New Thiazolidinone and Oxazolidinone Derived from Levofloxacin and Evaluation of Anti-Oxidant
by: Mustafa Moaied Rabeaa, et al.
Published: (2024-01-01)

Rethinking, reducing, and refining the classical oral tyramine challenge test of monoamine oxidase (MAO) inhibitors
by: Ewoud‐Jan vanHoogdalem, et al.
Published: (2023-10-01)

Synthesis and Structural Study of Amidrazone Derived Pyrrole-2,5-Dione Derivatives: Potential Anti-Inflammatory Agents
by: Renata Paprocka, et al.
Published: (2022-04-01)

Synthesis and Anti-Tuberculosis Activity of Substituted 3,4-(dicoumarin-3-yl)-2,5-diphenyl Furans and Pyrroles
by: Bhagwat Jadhav, et al.
Published: (2022-12-01)

STUDY MOLECULES DOCKING OF ALKALOIDS IN KRATOM ON SEROTONIN TRANSPORTER (SERT), NOREPINEPHRINE TRANSPORTER (NET), AND MONOAMINE OXIDASE (MAO)
by: Dandi Irawan, et al.
Published: (2023-12-01)

BASE-INDUCED C-5 EPIMERIZATION OF 4-METHYL-5-PHENYL OXAZOLIDINONES - CHIRAL AUXILIARIES DERIVED FROM NOREPHEDRINE AND NORPSEUDOEPHEDRINE
by: Davies, S, et al.
Published: (1993)

2-(2,5-Dimethoxyphenyl)pyrrole-3-carbonitrile
by: Yannic Grimm, et al.
Published: (2023-04-01)

1-(3,5-Dimethoxybenzyl)-1H-pyrrole
by: Wei Huang, et al.
Published: (2012-05-01)

Synthesis, Antibacterial and Anthelmintic Activity of Novel 3-(3-Pyridyl)-oxazolidinone-5-methyl Ester Derivatives
by: Bo Jin, et al.
Published: (2022-02-01)

Improved Gas Hydrate Kinetic Inhibition for 5‑Methyl-3-vinyl-2-oxazolidinone Copolymers and Synergists
by: Malcolm A. Kelland, et al.
Published: (2023-07-01)

Monoamine Oxidase (MAO) Is Expressed at the Level of Mitral Valve with Severe Regurgitation in Hypertrophic Obstructive Cardiomyopathy: A Case Report
by: Ana Lascu, et al.
Published: (2022-12-01)

Molecular and structural basis of anti-DNA antibody specificity for pyrrolated proteins
by: Yusuke Anan, et al.
Published: (2024-02-01)

Oxazolidinones as an Alternative in the Treatment of Multiresistant Staphylococcus Aureus
by: Maira Quiros Enríquez, et al.
Published: (2013-04-01)

Oxazolidinone Antibiotics: Chemical, Biological and Analytical Aspects
by: Claudia Foti, et al.
Published: (2021-07-01)

5-{2-[(2-Hydroxy-5-methylphenyl)(phenyl)methyleneamino]phenyliminomethyl}pyrrole-2-carbaldehyde
by: Ge Liu, et al.
Published: (2008-08-01)

Enantioselective Interactions of Anti-Infective 8-Aminoquinoline Therapeutics with Human Monoamine Oxidases A and B
by: Narayan D. Chaurasiya, et al.
Published: (2021-04-01)

Biological evaluation, molecular docking and DFT calculations of pyrrole-based derivatives as dual acting AChE/MAO-B inhibitors
by: Emilio Mateev, et al.
Published: (2023-10-01)

Design and synthesis of potential pyrrole-coupled carboxamide derivatives as an anti-superbug MRSA agent
by: Boobal Arasu Velu, et al.
Published: (2024-01-01)

Efficient fabrication of oxazolidinones for the carboxylative cyclization with carbon dioxide
by: Xin Yang, et al.
Published: (2023-08-01)

5,7-Dimethoxycoumarin ameliorates vincristine induced neuropathic pain: potential role of 5HT3 receptors and monoamines
by: Muhammad Usman, et al.
Published: (2023-10-01)

In Silico Evaluation and In Vitro Determination of Neuroprotective and MAO-B Inhibitory Effects of Pyrrole-Based Hydrazones: A Therapeutic Approach to Parkinson’s Disease
by: Magdalena Kondeva-Burdina, et al.
Published: (2022-12-01)

Flexibility in the partial reduction of 2,5-disubstituted pyrroles: application to the synthesis of DMDP.
by: Donohoe, T, et al.
Published: (2003)

(3,5-Dimethyl-1H-pyrrol-2-yl)(phenyl)methanone
by: Fengzhen Wang, et al.
Published: (2016-05-01)

Platelet Serotonin (5-HT) Concentration, Platelet Monoamine Oxidase B (MAO-B) Activity and <i>HTR2A</i>, <i>HTR2C</i>, and <i>MAOB</i> Gene Polymorphisms in Asthma
by: Marcela Konjevod, et al.
Published: (2023-05-01)

Optimization and Antibacterial Evaluation of Novel 3-(5-Fluoropyridine-3-yl)-2-oxazolidinone Derivatives Containing a Pyrimidine Substituted Piperazine
by: Xin Wang, et al.
Published: (2023-05-01)

Synthesis and Characterization of Novel Oxazolidinones Via Schiff Base Reactions
by: Obaid H.Abid, et al.
Published: (2013-11-01)

Synergistic Activity of Nitroimidazole-Oxazolidinone Conjugates against Anaerobic Bacteria
by: Zhijun Zhuang, et al.
Published: (2020-05-01)

Mao Mao : inside Gary's head
by: Chia, Gary Yew Hong
Published: (2019)

Direct routes to 5,15-diaryl-10,20-diethynyl porphyrins from pyrrole
by: Wilson, G, et al.
Published: (1996)

BF₃-promoted reactions of α-amino acetals with alkynes to 2,5-disubstituted pyrroles
by: Gao, Zhi-Yuan, et al.
Published: (2022)

rac-1-(4-tert-Butylphenyl)-5-ethyl-4-ferrocenyl-5-hydroxy-1H-pyrrol-2(5H)-one
by: Tobias Biletzki, et al.
Published: (2023-04-01)

Crystal structure of (Z)-2-(tert-butyl)-5-((5-(tert- butyl)-2H-pyrrol-2-ylidene)(mesityl)methyl)-1H-pyrrole, C26H34N2
by: Liu Yingfan, et al.
Published: (2022-10-01)

Antibacterial Properties and Computational Insights of Potent Novel Linezolid-Based Oxazolidinones
by: M. Shaheer Malik, et al.
Published: (2023-03-01)

Syntheses and Crystal Structures of Three Chiral Oxazolidinones with Different Ring Conformations
by: Ester Soru, et al.
Published: (2022-11-01)

COMPARISON OF THE CLINICAL ACTIVITY OF TWO OXAZOLIDINONES – LINEZOLID AND TEDIZOLIDE: UNJUSTIFIED EXPECTATIONS
by: N. V. Dmitrieva, et al.
Published: (2018-11-01)

Structural basis for PoxtA-mediated resistance to phenicol and oxazolidinone antibiotics
by: Caillan Crowe-McAuliffe, et al.
Published: (2022-04-01)