Functional Expression of Adenosine A<sub>3</sub> Receptor in Yeast Utilizing a Chimera with the A<sub>2A</sub>R C-Terminus
The adenosine A<sub>3</sub> receptor (A<sub>3</sub>R) is the only adenosine receptor subtype to be overexpressed in inflammatory and cancer cells and therefore is considered a novel and promising therapeutic target for inflammatory diseases and cancer. Heterologous expression...
Main Authors: | Abhinav R. Jain, Anne S. Robinson |
---|---|
Format: | Article |
Language: | English |
Published: |
MDPI AG
2020-06-01
|
Series: | International Journal of Molecular Sciences |
Subjects: | |
Online Access: | https://www.mdpi.com/1422-0067/21/12/4547 |
Similar Items
-
Allosteric Antagonism of the A<sub>2A</sub> Adenosine Receptor by a Series of Bitopic Ligands
by: Zhan-Guo Gao, et al.
Published: (2020-05-01) -
Identification of TSPAN4 as Novel Histamine H<sub>4</sub> Receptor Interactor
by: Xiaoyuan Ma, et al.
Published: (2021-07-01) -
Molecular Biophysics of Class A G Protein Coupled Receptors–Lipids Interactome at a Glance—Highlights from the A<sub>2A</sub> Adenosine Receptor
by: Efpraxia Tzortzini, et al.
Published: (2023-06-01) -
Two-Dimensional NMR Spectroscopy of the G Protein-Coupled Receptor A<sub>2A</sub>AR in Lipid Nanodiscs
by: Canyong Guo, et al.
Published: (2023-07-01) -
BRET-Based Biosensors to Measure Agonist Efficacies in Histamine H<sub>1</sub> Receptor-Mediated G Protein Activation, Signaling and Interactions with GRKs and β-Arrestins
by: Eléonore W. E. Verweij, et al.
Published: (2022-03-01)