Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Aryl Sulfonamides

Bibliographic Details
Main Authors: Sudarsana Reddy Vanga, Jonas Sävmarker, Leelee Ng, Mats Larhed, Mathias Hallberg, Johan Åqvist, Anders Hallberg, Siew Yeen Chai, Hugo Gutiérrez-de-Terán
Format: Article
Language:English
Published: American Chemical Society 2018-04-01
Series:ACS Omega
Online Access:http://dx.doi.org/10.1021/acsomega.8b00595
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author Sudarsana Reddy Vanga
Jonas Sävmarker
Leelee Ng
Mats Larhed
Mathias Hallberg
Johan Åqvist
Anders Hallberg
Siew Yeen Chai
Hugo Gutiérrez-de-Terán
author_facet Sudarsana Reddy Vanga
Jonas Sävmarker
Leelee Ng
Mats Larhed
Mathias Hallberg
Johan Åqvist
Anders Hallberg
Siew Yeen Chai
Hugo Gutiérrez-de-Terán
author_sort Sudarsana Reddy Vanga
collection DOAJ
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issn 2470-1343
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spelling doaj.art-bfde87a0178d46798e868c6357b433912022-12-22T00:30:03ZengAmerican Chemical SocietyACS Omega2470-13432018-04-01344509452110.1021/acsomega.8b00595Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Aryl SulfonamidesSudarsana Reddy Vanga0Jonas Sävmarker1Leelee Ng2Mats Larhed3Mathias Hallberg4Johan Åqvist5Anders Hallberg6Siew Yeen Chai7Hugo Gutiérrez-de-Terán8Department of Cell and Molecular Biology, BMC, Uppsala University, Uppsala, Sweden‡Department of Medicinal Chemistry, Uppsala University, BMC, Uppsala, SwedenBiomedicine Discovery Institute, Department of Physiology, Monash University, Clayton, Victoria, Australia‡Department of Medicinal Chemistry, Uppsala University, BMC, Uppsala, SwedenThe Beijer Laboratory, Department of Pharmaceutical Biosciences, Division of Biological Research on Drug Dependence, Uppsala University, BMC, Uppsala, SwedenDepartment of Cell and Molecular Biology, BMC, Uppsala University, Uppsala, Sweden‡Department of Medicinal Chemistry, Uppsala University, BMC, Uppsala, SwedenBiomedicine Discovery Institute, Department of Physiology, Monash University, Clayton, Victoria, AustraliaDepartment of Cell and Molecular Biology, BMC, Uppsala University, Uppsala, Swedenhttp://dx.doi.org/10.1021/acsomega.8b00595
spellingShingle Sudarsana Reddy Vanga
Jonas Sävmarker
Leelee Ng
Mats Larhed
Mathias Hallberg
Johan Åqvist
Anders Hallberg
Siew Yeen Chai
Hugo Gutiérrez-de-Terán
Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Aryl Sulfonamides
ACS Omega
title Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Aryl Sulfonamides
title_full Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Aryl Sulfonamides
title_fullStr Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Aryl Sulfonamides
title_full_unstemmed Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Aryl Sulfonamides
title_short Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Aryl Sulfonamides
title_sort structural basis of inhibition of human insulin regulated aminopeptidase irap by aryl sulfonamides
url http://dx.doi.org/10.1021/acsomega.8b00595
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