A Robust Bioassay of the Human Bradykinin B<sub>2</sub> Receptor That Extends Molecular and Cellular Studies: The Isolated Umbilical Vein
Bradykinin (BK) has various physiological and pathological roles. Medicinal chemistry efforts targeted toward the widely expressed BK B<sub>2</sub> receptor (B<sub>2</sub>R), a G-protein-coupled receptor, were primarily aimed at developing antagonists. The only B<sub>2&...
Main Authors: | François Marceau, Hélène Bachelard |
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Format: | Article |
Language: | English |
Published: |
MDPI AG
2021-02-01
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Series: | Pharmaceuticals |
Subjects: | |
Online Access: | https://www.mdpi.com/1424-8247/14/3/177 |
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