Hot-Melt Extruded Amorphous Solid Dispersion for Solubility, Stability, and Bioavailability Enhancement of Telmisartan

Telmisartan (TEL, an antihypertensive drug) belongs to Class II of the Biopharmaceutical Classification System (BCS) because of its poor aqueous solubility. In this study, we enhanced the solubility, bioavailability, and stability of TEL through the fabrication of TEL-loaded pH-modulated solid dispe...

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Xehetasun bibliografikoak
Egile Nagusiak: Bhupendra Raj Giri, Jaewook Kwon, Anh Q. Vo, Ajinkya M. Bhagurkar, Suresh Bandari, Dong Wuk Kim
Formatua: Artikulua
Hizkuntza:English
Argitaratua: MDPI AG 2021-01-01
Saila:Pharmaceuticals
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Sarrera elektronikoa:https://www.mdpi.com/1424-8247/14/1/73