Heterodimerization of Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Leads to Increased M2R Affinity and Selectivity

Bibliographic Details
Main Authors: Xueke She, Andrea Pegoli, Judith Mayr, Harald Hübner, Günther Bernhardt, Peter Gmeiner, Max Keller
Format: Article
Language:English
Published: American Chemical Society 2017-10-01
Series:ACS Omega
Online Access:http://dx.doi.org/10.1021/acsomega.7b01085
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author Xueke She
Andrea Pegoli
Judith Mayr
Harald Hübner
Günther Bernhardt
Peter Gmeiner
Max Keller
author_facet Xueke She
Andrea Pegoli
Judith Mayr
Harald Hübner
Günther Bernhardt
Peter Gmeiner
Max Keller
author_sort Xueke She
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issn 2470-1343
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spelling doaj.art-ccc71977ac8542fabfefb2480ed6e0de2022-12-21T23:56:05ZengAmerican Chemical SocietyACS Omega2470-13432017-10-012106741675410.1021/acsomega.7b01085Heterodimerization of Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Leads to Increased M2R Affinity and SelectivityXueke She0Andrea Pegoli1Judith Mayr2Harald Hübner3Günther Bernhardt4Peter Gmeiner5Max Keller6Institute of Pharmacy, Faculty of Chemistry and Pharmacy, University of Regensburg, Regensburg, GermanyInstitute of Pharmacy, Faculty of Chemistry and Pharmacy, University of Regensburg, Regensburg, GermanyInstitute of Pharmacy, Faculty of Chemistry and Pharmacy, University of Regensburg, Regensburg, GermanyDepartment of Chemistry and Pharmacy, Emil Fischer Center, Friedrich Alexander University, Erlangen, GermanyInstitute of Pharmacy, Faculty of Chemistry and Pharmacy, University of Regensburg, Regensburg, GermanyDepartment of Chemistry and Pharmacy, Emil Fischer Center, Friedrich Alexander University, Erlangen, GermanyInstitute of Pharmacy, Faculty of Chemistry and Pharmacy, University of Regensburg, Regensburg, Germanyhttp://dx.doi.org/10.1021/acsomega.7b01085
spellingShingle Xueke She
Andrea Pegoli
Judith Mayr
Harald Hübner
Günther Bernhardt
Peter Gmeiner
Max Keller
Heterodimerization of Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Leads to Increased M2R Affinity and Selectivity
ACS Omega
title Heterodimerization of Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Leads to Increased M2R Affinity and Selectivity
title_full Heterodimerization of Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Leads to Increased M2R Affinity and Selectivity
title_fullStr Heterodimerization of Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Leads to Increased M2R Affinity and Selectivity
title_full_unstemmed Heterodimerization of Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Leads to Increased M2R Affinity and Selectivity
title_short Heterodimerization of Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Leads to Increased M2R Affinity and Selectivity
title_sort heterodimerization of dibenzodiazepinone type muscarinic acetylcholine receptor ligands leads to increased m2r affinity and selectivity
url http://dx.doi.org/10.1021/acsomega.7b01085
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