Palladium-Catalyzed Benzodiazepines Synthesis

Palladium-Catalyzed Benzodiazepines Synthesis

This review is focused on palladium-catalyzed reactions as efficient strategies aimed at the synthesis of different classes of benzodiazepines. Several reaction typologies are reported including hydroamination, amination, C–H arylation, N-arylation, and the Buchwald–Hartwig reaction, depending on th...

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Bibliographic Details
Main Authors:	Michael S. Christodoulou, Egle M. Beccalli, Sabrina Giofrè
Format:	Article
Language:	English
Published:	MDPI AG 2020-06-01
Series:	Catalysts
Subjects:	Pd-catalysis benzodiazepine cyclization domino process intramolecular Buchwald–Hartwig N-arylation
Online Access:	https://www.mdpi.com/2073-4344/10/6/634

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