A speedy route to sterically encumbered, benzene-fused derivatives of privileged, naturally occurring hexahydropyrrolo[1,2-b]isoquinoline
A series of 15 benzene-fused hexahydropyrrolo[1,2-b]isoquinolonic acids with substantial degree of steric encumbrance has been prepared via a novel variant of the Castagnoli–Cushman reaction of homophthalic anhydride (HPA) and various indolenines. The employment of a special kind of a cyclic imine c...
Main Authors: | Olga Bakulina, Alexander Ivanov, Vitalii Suslonov, Dmitry Dar’in, Mikhail Krasavin |
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Format: | Article |
Language: | English |
Published: |
Beilstein-Institut
2017-07-01
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Series: | Beilstein Journal of Organic Chemistry |
Subjects: | |
Online Access: | https://doi.org/10.3762/bjoc.13.138 |
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